SCHEMBL4445648

SCHEMBL4445648

CCCc1cc2ccc(OC)cc2s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.49
BACE1 P56817 1/20 0.44
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
MAPT P10636 5/20 0.41
POLB P06746 1/20 0.41
PDK1 Q15118 1/20 0.41
APOBEC3A P31941 1/20 0.40
TSHR P16473 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
CYP2A6 P11509 1/20 0.40
PSMB8 P28062 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
KMT2A Q03164 2/20 0.38
HPGD P15428 2/20 0.38
ALDH1A1 P00352 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30416457 0.88 CA2 (0.50) CA2BACE1CYP1A2CYP3A4CYP2C19
SCHEMBL4440695 0.88 CA2 (0.44) CA2BACE1CYP1A2CYP3A4CYP2C19
SCHEMBL5243924 0.86 CA2 (0.51) CA2BACE1CYP1A2CYP3A4CYP2C19
SCHEMBL5553145 0.85 CA2 (0.48) CA2BACE1CYP1A2CYP3A4CYP2C19
SCHEMBL5553012 0.85 CA2 (0.48) CA2BACE1CYP1A2CYP3A4CYP2C19
SCHEMBL534427 0.81 CYP2A6 (0.53) CA2BACE1CYP1A2CYP3A4CYP2C19
SCHEMBL13632630 0.79 CA2 (0.48) CA2BACE1CYP1A2CYP3A4CYP2C19
SCHEMBL5557274 0.78 CA2 (0.51) CA2CYP1A2CYP3A4CYP2C19MAPT
SCHEMBL5557265 0.78 CA2 (0.51) CA2BACE1CYP1A2CYP3A4CYP2C19
SCHEMBL13632619 0.77 CA2 (0.41) CA2BACE1CYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7476691-B2 Sulfamate benzothiophene derivatives as steroid sulfatase inhibitors LABORATOIRE THERAMEX (MC) 2009-01-13 US disclosed