SCHEMBL4445888

SCHEMBL4445888

COC(=O)c1cc(Cl)c(OC)cc1O.O=C(O)c1cc(Cl)c(O)cc1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.49
HSP90AA1 P07900 4/20 0.44
HTT P42858 3/20 0.43
PYGL P06737 2/20 0.43
KDM4E B2RXH2 4/20 0.41
MAPT P10636 3/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
NPC1 O15118 3/20 0.41
HSD17B10 Q99714 2/20 0.41
MAPK1 P28482 1/20 0.41
NOD2 Q9HC29 1/20 0.41
RECQL P46063 2/20 0.41
HPGD P15428 2/20 0.41
LMNA P02545 1/20 0.41
CYP3A4 P08684 1/20 0.41
POLB P06746 2/20 0.41
ABL1 P00519 1/20 0.41
PKM P14618 1/20 0.41
BLM P54132 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2793251 0.89 GAA (0.58) GAAHTTKDM4EMAPTMEN1
SCHEMBL4177645 0.88 HTT (0.52) GAAHTTPYGLKDM4EMAPT
SCHEMBL2726967 0.84 CA12 (0.53) GAAHSP90AA1KDM4ELMNAPOLB
SCHEMBL30463099 0.84 CA12 (0.53) GAAHSP90AA1KDM4ELMNAPOLB
SCHEMBL1742880 0.83 GAA (0.68) GAAHSP90AA1HTTKDM4EMAPT
SCHEMBL1743592 0.81 ALDH1A1 (0.51) GAAHSP90AA1HTTKDM4EHSD17B10
SCHEMBL30912978 0.81 CA12 (0.57) GAAHTTKDM4EMAPTMEN1
SCHEMBL29046583 0.80 GAA (0.63) GAAHTTKDM4EMAPTMEN1
SCHEMBL3467699 0.79 NPC1 (0.54) GAAHTTKDM4EMAPTMEN1
SCHEMBL3461530 0.78 KDM4E (0.57) GAAHTTKDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069355-A1 NOVEL TRICYCLIC SPIROPIPERIDINE COMPOUNDS, THEIR SYNTHESIS AND THEIR USES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY AstraZeneca AB (SE) 2009-06-17 EP disclosed
WO-2008010765-A1 NOVEL TRICYCLIC SPIROPIPERIDINE COMPOUNDS, THEIR SYNTHESIS AND THEIR USES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY ASTRAZENECA AB (SE) 2008-01-24 WO disclosed