SCHEMBL4447770

SCHEMBL4447770

COc1cccc(-c2[c]nn[nH]2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DCUN1D1 Q96GG9 1/20 0.50
DYRK1A Q13627 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
GAA P10253 3/20 0.48
NOTUM Q6P988 2/20 0.47
NR1H2 P55055 1/20 0.47
NR1H3 Q13133 1/20 0.47
XDH P47989 1/20 0.47
NISCH Q9Y2I1 1/20 0.45
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2B6 P20813 2/20 0.43
CYP1A1 P04798 1/20 0.43
CYP2E1 P05181 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C8 P10632 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2A6 P11509 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL196765 0.73 CYP3A4 (0.73) DYRK1ACLK4GAANOTUMXDH
SCHEMBL29489425 0.73 CYP3A4 (0.73) DYRK1ACLK4GAANOTUMXDH
Ammonia Solution, Strong SCHEMBL27960505 0.71 CYP3A4 (0.70) DYRK1ACLK4GAANOTUMXDH
SCHEMBL29628977 0.71 CYP3A4 (0.77) DYRK1ACLK4GAANOTUMXDH
Hydrogen Sulfide SCHEMBL28640169 0.71 CYP3A4 (0.70) DYRK1ACLK4GAANOTUMXDH
SCHEMBL703677 0.70 DCUN1D1 (0.54) DCUN1D1DYRK1ACLK4GAANOTUM
SCHEMBL1180343 0.69 ABL1 (0.69) DYRK1ACLK4XDHCYP1A2CYP2C9
SCHEMBL4720179 0.69 ALDH1A1 (0.50) DCUN1D1GAAXDHMAPTSMN1; SMN2
SCHEMBL4053635 0.69 GAA (0.50) DCUN1D1DYRK1ACLK4GAANOTUM
SCHEMBL4041229 0.69 DCUN1D1 (0.52) DCUN1D1DYRK1ACLK4GAANOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2056844-A2 NOVEL MACROLIDES AND KETOLIDES HAVING ANTIMICROBIAL ACTIVITY Wockhardt Research Centre (IN) 2009-05-13 EP claimed
WO-2008023248-A2 NOVEL MACROLIDES AND KETOLIDES HAVING ANTIMICROBIAL ACTIVITY WOCKHARDT RESEARCH CENTRE (IN) 2008-02-28 WO claimed