SCHEMBL4447866

SCHEMBL4447866

CC(C)(C(N)=O)c1cc(N)ccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.42
TSHR P16473 2/20 0.42
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
NR1H4 Q96RI1 4/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
HSD17B10 Q99714 3/20 0.38
ALDH1A1 P00352 1/20 0.38
THRB P10828 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
CASP1 P29466 1/20 0.38
RECQL P46063 1/20 0.38
EPHX2 P34913 1/20 0.38
MAPK1 P28482 1/20 0.37
RIPK2 O43353 2/20 0.37
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4438664 0.86 CYP3A4 (0.42) CYP3A4TSHRMAPTKMT2ANR1H4
SCHEMBL19461805 0.77 GAA (0.48) TSHRMAPTKMT2AHSD17B10ALDH1A1
SCHEMBL1762358 0.77 TSHR (0.52) CYP3A4TSHRMAPTNR1H4CA1
SCHEMBL4440253 0.76 KMT2A (0.53) CYP3A4TSHRMAPTKMT2ANR1H4
SCHEMBL19815146 0.76 MAPT (0.53) MAPTKMT2AALDH1A1NPC1RAB9A
SCHEMBL28785557 0.73 CYP3A4 (0.48) CYP3A4TSHRMAPTNR1H4CA1
SCHEMBL1762437 0.73 TSHR (0.48) CYP3A4TSHRMAPTCA1CA2
SCHEMBL30707878 0.71 CYP3A4 (0.42) CYP3A4TSHRMAPTKMT2ACA1
SCHEMBL27176545 0.71 CYP3A4 (0.42) CYP3A4TSHRMAPTKMT2ACA1
SCHEMBL8443184 0.70 KMT2A (0.52) TSHRMAPTKMT2AEPHX2RIPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134676-A2 NOVEL BENZAMIDE DERIVATIVES AS MODULATORS OF THE FOLLICLE STIMULATING HORMONE Addex Pharma SA (CH) 2009-12-23 EP disclosed
WO-2008117175-A2 NOVEL BENZAMIDE DERIVATIVES AS MODULATORS OF THE FOLLICLE STIMULATING HORMONE ADDEX PHARMA SA (CH) 2008-10-02 WO disclosed