SCHEMBL4438664

SCHEMBL4438664

CC(C)(C(N)=O)c1ccc(N)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
TSHR P16473 2/20 0.42
NR1H4 Q96RI1 4/20 0.42
HSD17B10 Q99714 3/20 0.42
ALDH1A1 P00352 1/20 0.42
THRB P10828 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
CASP1 P29466 1/20 0.42
RECQL P46063 1/20 0.42
EPHX2 P34913 1/20 0.40
MAPT P10636 3/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.38
HSD11B1 P28845 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
JAK2 O60674 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4447866 0.86 CYP3A4 (0.42) CYP3A4CA1CA2TSHRNR1H4
SCHEMBL19461805 0.77 GAA (0.48) TSHRHSD17B10ALDH1A1HPGDCASP1
SCHEMBL3781096 0.77 CYP3A4 (0.52) CYP3A4CA1CA2TSHRNR1H4
SCHEMBL8128654 0.77 CYP3A4 (0.52) CYP3A4CA1CA2TSHRNR1H4
SCHEMBL2817983 0.76 KMT2A (0.56) NR1H4HSD17B10ALDH1A1MAPTKMT2A
SCHEMBL19815146 0.76 MAPT (0.53) ALDH1A1MAPTKMT2A
SCHEMBL27776101 0.75 CYP3A4 (0.50) CYP3A4CA1CA2TSHRNR1H4
SCHEMBL10781060 0.71 CYP3A4 (0.42) CYP3A4CA1CA2TSHRNR1H4
SCHEMBL2817651 0.71 NR1H4 (0.44) CYP3A4CA1CA2TSHRNR1H4
SCHEMBL4573292 0.70 ADRB1 (0.54) CYP3A4TSHRHSD17B10ALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134676-A2 NOVEL BENZAMIDE DERIVATIVES AS MODULATORS OF THE FOLLICLE STIMULATING HORMONE Addex Pharma SA (CH) 2009-12-23 EP disclosed
WO-2008117175-A2 NOVEL BENZAMIDE DERIVATIVES AS MODULATORS OF THE FOLLICLE STIMULATING HORMONE ADDEX PHARMA SA (CH) 2008-10-02 WO disclosed