SCHEMBL4447953

SCHEMBL4447953

CSCCC1CC(c2cccc(C(F)(F)F)c2)N(c2ccc(Oc3ccc(Cl)cc3)cc2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CETP P11597 1/20 0.36
CNR1 P21554 3/20 0.36
CNR2 P34972 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
NPBWR1 P48145 2/20 0.34
MCHR1 Q99705 1/20 0.34
SCN9A Q15858 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
DRD2 P14416 1/20 0.33
MC4R P32245 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3592600 1.00 HTT (0.38) HTTMEN1KMT2ACYP1A2CYP3A4
SCHEMBL15181797 0.91 HTT (0.39) HTTMEN1KMT2ACYP1A2CYP3A4
SCHEMBL15181817 0.90 HTT (0.39) HTTMEN1KMT2ACYP1A2CYP3A4
SCHEMBL3598463 0.89 HTT (0.41) HTTMEN1KMT2ACYP1A2CYP3A4
SCHEMBL3591231 0.89 HTT (0.41) HTTMEN1KMT2ACYP1A2CYP3A4
SCHEMBL4439759 0.89 HTT (0.41) HTTMEN1KMT2ACYP1A2CYP3A4
SCHEMBL3585646 0.88 HTT (0.37) HTTMEN1KMT2ACYP1A2CYP3A4
SCHEMBL3586449 0.88 HTT (0.37) HTTMEN1KMT2ACYP1A2CYP3A4
SCHEMBL4437675 0.88 HTT (0.37) HTTMEN1KMT2ACYP1A2CYP3A4
SCHEMBL3591435 0.88 HTT (0.40) HTTMEN1KMT2ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121598-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2009-11-25 EP disclosed
WO-2008076754-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-06-26 WO disclosed