SCHEMBL4448448

SCHEMBL4448448

CCCCC(=O)C(Cc1ccc(-c2ccccc2)c(C#N)c1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.41
TSHR P16473 1/20 0.40
MME P08473 4/20 0.39
CTSB P07858 1/20 0.39
SLC22A12 Q96S37 1/20 0.39
XDH P47989 2/20 0.39
ITGB1 P05556 1/20 0.39
ITGA4 P13612 1/20 0.39
ACE P12821 3/20 0.38
LTB4R2 Q9NPC1 1/20 0.38
CPA1 P15085 1/20 0.38
ACE2 Q9BYF1 1/20 0.38
GRM5 P41594 1/20 0.38
PTPN1 P18031 1/20 0.38
DGAT1 O75907 1/20 0.37
WNT3A P56704 1/20 0.37
MRE11 P49959 1/20 0.37
FFAR1 O14842 1/20 0.36
AKR1B1 P15121 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4018176 0.93 SLC22A12 (0.42) CYP19A1MMESLC22A12XDHITGB1
SCHEMBL4018178 0.93 SLC22A12 (0.42) CYP19A1MMESLC22A12XDHITGB1
SCHEMBL2572010 0.87 MME (0.52) TSHRMMEITGB1ITGA4ACE
SCHEMBL9710320 0.84 MME (0.51) TSHRMMEITGB1ITGA4ACE
SCHEMBL9448762 0.84 MMP8 (0.41) CYP19A1MMEXDHGRM5DGAT1
SCHEMBL9710219 0.83 MME (0.50) TSHRMMEITGB1ITGA4ACE
SCHEMBL9710577 0.83 MME (0.50) TSHRMMEITGB1ITGA4ACE
SCHEMBL8317308 0.80 MME (0.54) MMEITGB1ITGA4PTPN1FFAR1
SCHEMBL27792670 0.80 MMP8 (0.46) CYP19A1XDHGRM5DGAT1WNT3A
SCHEMBL4321176 0.78 KMT2A (0.39) TSHRMMECTSBACELTB4R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed