SCHEMBL4448751

SCHEMBL4448751

O=C1c2cccc3cccc(c23)C(=O)N1CCCCl

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HEXA P06865 6/20 0.71
HEXB P07686 6/20 0.71
KMT2A Q03164 2/20 0.65
POLB P06746 2/20 0.65
MEN1 O00255 1/20 0.65
NR1I2 O75469 1/20 0.65
AHR P35869 1/20 0.65
RAD52 P43351 1/20 0.65
RCE1 Q9Y256 1/20 0.65
SIRT1 Q96EB6 3/20 0.63
OGA O60502 1/20 0.63
CYP3A4 P08684 1/20 0.61
NFKB1 P19838 1/20 0.61
HSD17B10 Q99714 1/20 0.61
KDM4E B2RXH2 2/20 0.60
ALDH1A1 P00352 2/20 0.60
SMN1; SMN2 Q16637 2/20 0.60
HPGD P15428 1/20 0.60
HK1 P19367 1/20 0.60
APEX1 P27695 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22683219 0.97 HEXA (0.73) HEXAHEXBKMT2APOLBMEN1
SCHEMBL9034219 0.89 HEXA (0.69) HEXAHEXBKMT2APOLBMEN1
SCHEMBL9626265 0.89 HEXA (0.83) HEXAHEXBKMT2APOLBMEN1
SCHEMBL9625779 0.87 HEXA (0.81) HEXAHEXBKMT2APOLBMEN1
SCHEMBL9625395 0.87 HEXA (0.81) HEXAHEXBKMT2APOLBMEN1
SCHEMBL9625535 0.87 HEXA (0.81) HEXAHEXBKMT2APOLBMEN1
SCHEMBL9625518 0.87 HEXA (0.81) HEXAHEXBKMT2APOLBMEN1
SCHEMBL21450705 0.84 HEXA (0.73) HEXAHEXBKMT2APOLBMEN1
SCHEMBL31622484 0.83 MAPT (0.62) KMT2AMEN1SMN1; SMN2MAPTRAB9A
SCHEMBL5312972 0.83 MAPT (0.62) KMT2AMEN1SMN1; SMN2MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118065-B1 Substituted 1H-benz[de]isoquinoline-1,3-diones COUNCIL SCIENT IND RES (IN) 2013-08-14 EP disclosed
EP-2118065-A1 NOVEL SUBSTITUTED 1H-BENZ ÝDE¨ISOQUINOLINE-1, 3 -DIONES Council of Scientific & Industrial Research (IN) 2009-11-18 EP disclosed
WO-2008084496-A1 NOVEL SUBSTITUTED 1H-BENZ [DE] ISOQUINOLINE-1, 3 -DIONES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2008-07-17 WO disclosed