SCHEMBL4449200

SCHEMBL4449200

COC(=O)[C@@H](N)COCc1ccccc1.NC(=O)c1cnc(C(N)=O)cn1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC1A1 P43005 1/20 0.46
P4HTM Q9NXG6 1/20 0.45
LTA4H P09960 3/20 0.45
CNR1 P21554 1/20 0.44
SIRT6 Q8N6T7 1/20 0.40
GHSR Q92847 2/20 0.39
TACR1 P25103 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL589861 1.00 SLC1A1 (0.46) SLC1A1P4HTMLTA4HCNR1SIRT6
SCHEMBL4441919 0.87 SLC1A1 (0.57) SLC1A1P4HTMLTA4HCNR1TACR1
SCHEMBL2059074 0.87 SLC1A1 (0.57) SLC1A1LTA4HTACR1
SCHEMBL2389104 0.87 SLC1A1 (0.57) SLC1A1LTA4HTACR1
SCHEMBL1279255 0.87 SLC1A1 (0.57) SLC1A1LTA4HTACR1
Hydrochloric Acid SCHEMBL5487502 0.86 SLC1A1 (0.56) SLC1A1LTA4HTACR1
Hydrochloric Acid SCHEMBL5487507 0.86 SLC1A1 (0.56) SLC1A1LTA4HTACR1
Hydrochloric Acid SCHEMBL29886043 0.86 SLC1A1 (0.56) SLC1A1LTA4HTACR1
Hydrochloric Acid SCHEMBL5926216 0.78 SLC1A1 (0.48) SLC1A1LTA4H
SCHEMBL24103465 0.76 MAPT (0.52) SLC1A1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029554-B1 PYRAZINE DERIVATIVES AND USES THEREOF IN RENAL MONITORING MEDIBEACON LLC (US) 2014-03-19 EP disclosed
EP-2029554-A1 PYRAZINE DERIVATIVES AND USES THEREOF IN RENAL MONITORING Mallinckrodt, Inc. (US) 2009-03-04 EP disclosed
WO-2007149479-A1 PYRAZINE DERIVATIVES AND USES THEREOF IN RENAL MONITORING MALLINCKRODT INC. (US) 2007-12-27 WO disclosed