SCHEMBL4450897

SCHEMBL4450897

Clc1ccccc1N1CCN(CCCCOc2ccn3nccc3c2)CC1.O=[N+]([O-])c1cccc(N2CCN(CCCCOc3ccn4nccc4c3)CC2)c1

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 19/20 0.69
DRD4 P21917 19/20 0.69
DRD3 P35462 19/20 0.69
HTR2A P28223 16/20 0.59
DRD1 P21728 15/20 0.59
DRD5 P21918 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3615018 0.93 DRD2 (0.60) DRD2DRD4DRD3HTR2ADRD1
SCHEMBL3612201 0.86 DRD2 (0.86) DRD2DRD4DRD3HTR2ADRD1
SCHEMBL3615769 0.83 DRD2 (0.80) DRD2DRD4DRD3HTR2ADRD1
SCHEMBL3615538 0.82 DRD3 (1.00) DRD2DRD4DRD3HTR2ADRD1
SCHEMBL4441975 0.82 DRD2 (0.73) DRD2DRD4DRD3HTR2ADRD1
SCHEMBL3611425 0.79 DRD2 (0.93) DRD2DRD4DRD3HTR2ADRD1
SCHEMBL3603446 0.78 DRD3 (0.66) DRD2DRD4DRD3HTR2ADRD1
SCHEMBL28490438 0.77 DRD2 (0.66) DRD2DRD4DRD3HTR2ADRD1
SCHEMBL3611604 0.77 DRD2 (0.70) DRD2DRD4DRD3HTR2ADRD1
SCHEMBL3610425 0.76 DRD2 (0.65) DRD2DRD4DRD3HTR2ADRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137185-A2 INDOLIZINES AND AZA-ANALOG DERIVATIVES THEREOF AS CNS ACTIVE COMPOUNDS Gmeiner, Dr. Peter (DE) 2009-12-30 EP disclosed
WO-2008113559-A2 INDOLIZINES AND AZA-ANALOG DERIVATIVES THEREOF AS CNS ACTIVE COMPOUNDS SCHWARZ PHARMA AG (DE) 2008-09-25 WO disclosed