SCHEMBL4450940

SCHEMBL4450940

CCCc1nc(C(Br)Br)n(-c2ccc(OC)cc2)c(=O)c1Cc1ccccc1-c1ccccc1C#N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 5/20 0.41
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
CYP3A4 P08684 3/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
F10 P00742 1/20 0.36
NPBWR1 P48145 1/20 0.36
ALDH1A1 P00352 6/20 0.35
TSHR P16473 2/20 0.35
KDM4E B2RXH2 1/20 0.34
MAPT P10636 2/20 0.34
RXFP1 Q9HBX9 1/20 0.34
BACE1 P56817 1/20 0.34
APLNR P35414 1/20 0.34
TDP2 O95551 1/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1894600 0.89 PDE10A (0.40) PDE10AMEN1KMT2ACYP3A4CYP2C9
SCHEMBL4450943 0.86 CYP3A4 (0.39) PDE10AMEN1KMT2ACYP3A4CYP2C9
SCHEMBL4016370 0.80 F10 (0.38) PDE10AMEN1KMT2ACYP3A4CYP2C9
SCHEMBL1891376 0.80 PDE10A (0.40) PDE10AMEN1KMT2ACYP3A4CYP2C9
SCHEMBL12994037 0.80 PDE10A (0.40) PDE10AMEN1KMT2ACYP3A4CYP2C9
SCHEMBL4013362 0.78 MAPK1 (0.37) PDE10ACYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL13625902 0.78 ALDH1A1 (0.41) PDE10AMEN1KMT2ACYP3A4CYP2C9
SCHEMBL1892239 0.78 F10 (0.47) PDE10AMEN1KMT2ACYP3A4CYP2C9
SCHEMBL1895965 0.76 F10 (0.43) PDE10AMEN1KMT2ACYP3A4CYP2C9
SCHEMBL4013013 0.76 PDE10A (0.43) PDE10AMEN1KMT2ACYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed