SCHEMBL4452346

SCHEMBL4452346

Cc1ccc(C)n1-c1c[nH]nc1C(=O)O.Nc1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MYC P01106 10/20 0.42
NR4A1 P22736 3/20 0.36
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
LMNA P02545 3/20 0.35
MAPT P10636 3/20 0.35
NOTUM Q6P988 1/20 0.35
HAO2 Q9NYQ3 1/20 0.35
ALOX15 P16050 2/20 0.35
MEN1 O00255 1/20 0.35
THRB P10828 1/20 0.35
KMT2A Q03164 1/20 0.35
CASP1 P29466 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ESR1 P03372 1/20 0.35
PTPN7 P35236 1/20 0.35
HSD17B10 Q99714 1/20 0.35
AXL P30530 1/20 0.35
PTPN1 P18031 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2802546 0.86 MYC (0.53) MYCNR4A1KDM4EALDH1A1MAPT
SCHEMBL956958 0.77 CNR1 (0.47) KDM4EALDH1A1LMNAMAPTALOX15
SCHEMBL4343632 0.73 LRRK2 (0.36) ALDH1A1HAO2
SCHEMBL3937442 0.68 CFTR (0.35) ALOX15CASP1ESR1HSD17B10
SCHEMBL4442926 0.68 CDK2 (0.44) ALDH1A1LMNAMAPTALOX15MEN1
SCHEMBL4450271 0.68 HDAC1 (0.53) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL3939770 0.67 KDR (0.43) KDM4EMAPTMEN1KMT2ASMN1; SMN2
SCHEMBL1776218 0.65 CA12 (0.45) HAO2
SCHEMBL3979218 0.65
SCHEMBL15668778 0.62 MYC (0.68) MYCNR4A1KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049106-A2 PHARMACEUTICAL COMBINATIONS Astex Therapeutics Limited (GB) 2009-04-22 EP disclosed
WO-2008007113-A2 PHARMACEUTICAL COMBINATIONS ASTEX THERAPEUTICS LIMITED (GB) 2008-01-17 WO disclosed