SCHEMBL4452628

SCHEMBL4452628

O=c1cccc2ccccc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.47
ALOX12 P18054 1/20 0.47
GSTP1 P09211 1/20 0.46
GRIN2D O15399 1/20 0.44
GRIN3B O60391 1/20 0.44
GRIN1 Q05586 1/20 0.44
GRIN2A Q12879 1/20 0.44
GRIN2B Q13224 1/20 0.44
GRIN2C Q14957 1/20 0.44
GRIN3A Q8TCU5 1/20 0.44
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
CYP1A2 P05177 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HSD17B10 Q99714 2/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5243070 0.97 CYP2A6 (0.44) CYP2A6ALOX12GSTP1GRIN2DGRIN3B
Anthracene SCHEMBL5713428 0.73 CYP2A6 (0.73) CYP2A6ALOX12GSTP1CES2CES1
Naphthalene SCHEMBL28219404 0.73 CYP2A6 (0.73) CYP2A6ALOX12GSTP1GRIN2DGRIN3B
Naphthalene SCHEMBL27886370 0.73 CYP2A6 (0.73) CYP2A6ALOX12GSTP1GRIN2DGRIN3B
Anthracene SCHEMBL3187575 0.73 CYP2A6 (0.73) CYP2A6ALOX12GSTP1CES2CES1
SCHEMBL7905240 0.73 GSTP1 (0.48) CYP2A6ALOX12GSTP1GRIN2DGRIN3B
SCHEMBL6302567 0.71 CYP2A6 (0.57) CYP2A6ALOX12GSTP1CES2CES1
SCHEMBL29538674 0.71 CYP2A6 (0.57) CYP2A6ALOX12GSTP1CES2CES1
Anthracene SCHEMBL17912426 0.70 CYP2A6 (0.67) CYP2A6ALOX12CES2CES1CYP1A2
SCHEMBL5574323 0.70 CYP2A6 (0.54) CYP2A6ALOX12CYP1A2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2131657-A1 SUBSTITUTED BENZODIAZEPINONES, BENZOXAZEPINONES AND BENZOTHIAZEPINONES AS SODIUM CHANNEL BLOCKERS Merck & Co., Inc. (US) 2009-12-16 EP disclosed
WO-2008106077-A1 SUBSTITUTED BENZODIAZEPINONES, BENZOXAZEPINONES AND BENZOTHIAZEPINONES AS SODIUM CHANNEL BLOCKERS MERCK & CO., INC. (US) 2008-09-04 WO disclosed