SCHEMBL4453321

SCHEMBL4453321

NCCCC1COCCO1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.44
CHRM4 P08173 1/20 0.44
CHRM5 P08912 1/20 0.44
CHRM3 P20309 1/20 0.44
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
THRB P10828 1/20 0.36
EPHX1 P07099 1/20 0.33
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
KEAP1 Q14145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9557434 0.94 CHRM2 (0.42) CHRM2CHRM4CHRM5CHRM3ALDH1A1
SCHEMBL20367468 0.92 CHRM2 (0.39) CHRM2CHRM4CHRM5CHRM3ALDH1A1
SCHEMBL4445808 0.86
SCHEMBL21766160 0.86
SCHEMBL8084940 0.84 CHRM2 (0.45) CHRM2CHRM4CHRM5CHRM3ALDH1A1
SCHEMBL8084905 0.84 CHRM2 (0.45) CHRM2CHRM4CHRM5CHRM3ALDH1A1
SCHEMBL4578897 0.84 CHRM2 (0.45) CHRM2CHRM4CHRM5CHRM3ALDH1A1
SCHEMBL10197453 0.81
SCHEMBL25336760 0.78 CHRM2 (0.44) CHRM2CHRM4CHRM5CHRM3ALDH1A1
SCHEMBL4667952 0.78 CHRM2 (0.44) CHRM2CHRM4CHRM5CHRM3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819000-B1 NODULISPORIC ACID DERIVATIVES MERCK & CO INC (US) 2009-07-08 EP disclosed
EP-0819000-A4 NODULISPORIC ACID DERIVATIVES MERCK & CO INC (US) 2001-04-11 EP disclosed
US-5962499-A ACARICIDAL, ANTIPARASITIC, INSECTICIDAL AND ANTHELMINTIC AGENTS MERCK & CO., INC. (US) 1999-10-05 US disclosed
EP-0819000-A1 NODULISPORIC ACID DERIVATIVES Merck & Co., Inc. (US) 1998-01-21 EP disclosed
WO-1996029073-A1 NODULISPORIC ACID DERIVATIVES MERCK & CO., INC. (US) 1996-09-26 WO disclosed