SCHEMBL4455470

SCHEMBL4455470

CC(C)N1CCN(c2ncc(C(N)=O)cn2)CC1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 13/20 0.52
PTPN11 Q06124 1/20 0.48
OGA O60502 2/20 0.46
HDAC3 O15379 3/20 0.45
HDAC1 Q13547 3/20 0.45
HDAC2 Q92769 3/20 0.45
HDAC8 Q9BY41 3/20 0.45
HDAC4 P56524 2/20 0.45
HDAC7 Q8WUI4 2/20 0.45
HDAC10 Q969S8 2/20 0.45
HDAC11 Q96DB2 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
HDAC9 Q9UKV0 2/20 0.45
HDAC5 Q9UQL6 2/20 0.45
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28373607 0.82 HDAC3 (0.56) HDAC3HDAC1HDAC2HDAC8HDAC4
SCHEMBL23988327 0.82 OGA (0.44) HRH3PTPN11OGAHDAC3HDAC1
SCHEMBL23251484 0.82 OGA (0.44) HRH3PTPN11OGAHDAC3HDAC1
SCHEMBL4467331 0.81 HRH3 (0.69) HRH3OGA
SCHEMBL20917117 0.80 POLB (0.50) PTPN11HDAC3HDAC1HDAC2HDAC8
SCHEMBL24126684 0.79 HRH3 (0.44) HRH3OGAHDAC3HDAC1HDAC2
SCHEMBL4790004 0.78 POLB (0.49) PTPN11HDAC6POLB
SCHEMBL1126338 0.78 OGA (0.53) HRH3PTPN11OGA
SCHEMBL4456976 0.78 PTPN11 (0.48) HRH3PTPN11HDAC3HDAC1HDAC2
SCHEMBL63785 0.77 OGA (0.57) HRH3PTPN11OGAHDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009141386-A1 DERIVATIVES OF QUINOLINES AND QUINOXALINES AS PROTEIN TYROSINE KINASE INHIBITORS NOVARTIS AG (CH) 2009-11-26 WO disclosed