SCHEMBL4467331

SCHEMBL4467331

CC(C)N1CCN(c2ccc(C(N)=O)cn2)CC1

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 14/20 0.69
SMO Q99835 1/20 0.52
OPRM1 P35372 1/20 0.51
OPRK1 P41145 1/20 0.51
PARP1 P09874 1/20 0.50
OGA O60502 1/20 0.50
UBE2T Q9NPD8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30109094 0.87 HRH3 (0.69) HRH3SMOOGA
SCHEMBL7535374 0.86 HRH3 (0.55) HRH3OGA
SCHEMBL1860307 0.84 ALDH1A1 (0.60) HRH3
SCHEMBL7530613 0.84 HRH3 (0.54) HRH3OGA
Potassium Ion SCHEMBL7529500 0.84 HRH3 (0.54) HRH3OGA
SCHEMBL4460927 0.84 RAB9A (0.56) HRH3SMOOPRM1OPRK1PARP1
SCHEMBL12159827 0.83 NPC1 (0.55) HRH3OGAUBE2T
SCHEMBL14844055 0.83 HRH3 (1.00) HRH3
SCHEMBL31061451 0.83 HRH3 (1.00) HRH3
SCHEMBL14844995 0.83 HRH3 (1.00) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009141386-A1 DERIVATIVES OF QUINOLINES AND QUINOXALINES AS PROTEIN TYROSINE KINASE INHIBITORS NOVARTIS AG (CH) 2009-11-26 WO disclosed