SCHEMBL4456449

SCHEMBL4456449

CCOc1ccc(C(=O)O)cc1.O=[N+]([O-])c1ccc2cccnc2c1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.50
KMT2A Q03164 1/20 0.50
PLA2G4B P0C869 1/20 0.47
KDM4E B2RXH2 4/20 0.45
LMNA P02545 4/20 0.45
HTT P42858 3/20 0.45
L3MBTL1 Q9Y468 3/20 0.45
ADAMTS5 Q9UNA0 2/20 0.45
CCR6 P51684 1/20 0.45
ALDH1A1 P00352 4/20 0.45
MAPT P10636 4/20 0.45
GRK6 P43250 1/20 0.45
RCE1 Q9Y256 3/20 0.44
HSP90AA1 P07900 2/20 0.44
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4461356 0.92 PLA2G4B (0.51) PLA2G4BKDM4EALDH1A1MAPTHSP90AA1
SCHEMBL4462764 0.92 PLA2G4B (0.46) KMT2APLA2G4BKDM4ELMNAHTT
SCHEMBL4462759 0.92 PLA2G4B (0.46) KMT2APLA2G4BKDM4ELMNAHTT
SCHEMBL4465726 0.89 KMT2A (0.46) POLBKMT2AKDM4ELMNAHTT
SCHEMBL4461920 0.87 FEN1 (0.55) KMT2AKDM4ELMNAHTTL3MBTL1
SCHEMBL4461928 0.87 FEN1 (0.55) KMT2AKDM4ELMNAHTTL3MBTL1
SCHEMBL4458670 0.86 MAPT (0.51) KMT2AKDM4ELMNAHTTL3MBTL1
Benzoic Acid SCHEMBL4470207 0.85 ALDH1A1 (0.54) POLBKMT2AKDM4ELMNAHTT
Benzoic Acid SCHEMBL4470216 0.85 ALDH1A1 (0.54) POLBKMT2AKDM4ELMNAHTT
4-Nitrobenzoic Acid SCHEMBL4454979 0.84 KDR (0.54) KMT2AKDM4ELMNAHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009140215-A2 METHOD FOR TREATING DRUG-RESISTANT BACTERIAL AND OTHER INFECTIONS WITH CLIOQUINOL, PHANQUINONE, AND RELATED COMPOUNDS GERAGHTY, ERIN (US) 2009-11-19 WO claimed
WO-2009140215-A2 METHOD FOR TREATING DRUG-RESISTANT BACTERIAL AND OTHER INFECTIONS WITH CLIOQUINOL, PHANQUINONE, AND RELATED COMPOUNDS GERAGHTY, ERIN (US) 2009-11-19 WO disclosed