SCHEMBL4458826

SCHEMBL4458826

CC(C)c1cc(-c2c(N)nc(N)nc2N)n[nH]1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.46
TP53 P04637 7/20 0.41
MAPT P10636 6/20 0.41
AURKA O14965 2/20 0.40
PDPK1 O15530 2/20 0.40
TGFBR1 P36897 2/20 0.40
AURKB Q96GD4 2/20 0.40
DHFR P00374 1/20 0.39
SLC2A1 P11166 1/20 0.39
HCAR3 P49019 1/20 0.39
POLB P06746 2/20 0.38
RAF1 P04049 3/20 0.35
IKBKB O14920 1/20 0.33
BRAF P15056 1/20 0.32
COMT P21964 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4463005 0.78 HCAR2 (0.42) HCAR2TP53MAPTDHFRPOLB
SCHEMBL4458831 0.70 HCAR2 (0.49) HCAR2AURKAPDPK1TGFBR1AURKB
SCHEMBL1269500 0.69
SCHEMBL20928952 0.68 HCAR2 (0.45) HCAR2TP53MAPTHCAR3POLB
Hydrochloric Acid SCHEMBL21929877 0.67 HCAR2 (0.47) HCAR2TP53MAPTHCAR3
SCHEMBL2375615 0.66 TP53 (0.63) HCAR2TP53MAPTAURKBPOLB
SCHEMBL19400917 0.65
SCHEMBL19806475 0.64 CCR1 (0.53) HCAR2TP53MAPTPOLBRAF1
SCHEMBL14373074 0.64 SMN1; SMN2 (0.54) HCAR2TP53MAPTPOLB
SCHEMBL24120012 0.64 MAPT (0.51) HCAR2TP53MAPTHCAR3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed