SCHEMBL4463005

SCHEMBL4463005

CC(C)c1cc(-c2cnc(N)nc2N)n[nH]1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.42
TP53 P04637 4/20 0.41
MAPT P10636 3/20 0.41
DHFR P00374 5/20 0.41
POLB P06746 1/20 0.37
P2RX3 P56373 4/20 0.37
P2RX2 Q9UBL9 4/20 0.37
PIK3CA P42336 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30065933 0.80 NPC1 (0.50) HCAR2DHFRPIK3CA
SCHEMBL3663141 0.80 NPC1 (0.50) HCAR2DHFRPIK3CA
SCHEMBL29528815 0.78 DHFR (0.39) DHFRP2RX3P2RX2PIK3CA
SCHEMBL4458826 0.78 HCAR2 (0.46) HCAR2TP53MAPTDHFRPOLB
SCHEMBL4608258 0.76 DHFR (0.46) DHFRP2RX3P2RX2
SCHEMBL4457723 0.72 HCAR2 (0.43) HCAR2MAPTDHFRPIK3CA
Maleic Acid SCHEMBL28774616 0.70 DHFR (0.35) DHFRP2RX3P2RX2
SCHEMBL27976878 0.70 MKNK1 (0.35) HCAR2MAPTDHFRPIK3CA
SCHEMBL28664537 0.70 MKNK1 (0.40) HCAR2MAPTDHFRPIK3CA
SCHEMBL28814166 0.69 PIK3CA (0.37) DHFRPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed