SCHEMBL4459219

SCHEMBL4459219

O=C(NS(=O)(=O)c1ccc(F)cc1)c1ccc(-n2cnc3c(NC4CC4)nc(C(F)(F)F)nc32)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.40
CHEK1 O14757 1/20 0.40
NTRK1 P04629 1/20 0.40
MET P08581 1/20 0.40
PIM1 P11309 1/20 0.40
LTK P29376 1/20 0.40
GRK5 P34947 1/20 0.40
MAP2K2 P36507 1/20 0.40
CDK8 P49336 1/20 0.40
NEK2 P51955 1/20 0.40
LIMK1 P53667 1/20 0.40
TYRO3 Q06418 1/20 0.40
MAP4K2 Q12851 1/20 0.40
DYRK1A Q13627 1/20 0.40
AURKB Q96GD4 1/20 0.40
GRM1 Q13255 1/20 0.38
PTGS1 P23219 3/20 0.37
MCHR1 Q99705 1/20 0.37
TTK P33981 1/20 0.37
KDM1A O60341 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3146016 0.94 CHEK1 (0.36) PTGS2CHEK1NTRK1METPIM1
SCHEMBL3137695 0.92 TLR7 (0.39) TTKKDM1ASRCALKBH2ALKBH5
SCHEMBL3142068 0.90 YTHDC1 (0.38) PTGS2CHEK1NTRK1METPIM1
SCHEMBL3138810 0.87 TTK (0.38) CHEK1TTKSRC
SCHEMBL3141165 0.85 TTK (0.39) TYRO3TTKSRC
SCHEMBL3142034 0.85 GRM1 (0.46) NTRK1GRM1TP53
SCHEMBL3141046 0.84 YTHDC1 (0.41) PTGS2PTGS1SRCBCL2L1MCL1
SCHEMBL3137890 0.82 TLR7 (0.42) DYRK1A
SCHEMBL3145999 0.80 YTHDC1 (0.37) SRC
SCHEMBL3141117 0.80 YTHDC1 (0.39) TTKSRCEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009067607-A2 COMBINATIONS OF PDE4 INHIBITORS AND ANTIPSYCHOTICS FOR THE TREATMENT OF PSYCHOTIC DISORDERS MEMORY PHARMACEUTICALS CORPORATION (US) 2009-05-28 WO disclosed