SCHEMBL4459446

SCHEMBL4459446

CS(=O)(=O)c1ccc(Oc2ncnc3c2cnn3C2CCN(C(=O)O)CC2)cc1F

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.62
CYP2C9 P11712 2/20 0.50
GPR119 Q8TDV5 15/20 0.43
KCNH2 Q12809 1/20 0.41
BTK Q06187 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1128606 0.90 CYP3A4 (0.78) CYP3A4CYP2C9GPR119
SCHEMBL1128382 0.90 CYP3A4 (0.63) CYP3A4CYP2C9GPR119KCNH2
SCHEMBL1128845 0.86 CYP3A4 (0.55) CYP3A4CYP2C9GPR119KCNH2
SCHEMBL2019784 0.86 CYP3A4 (0.79) CYP3A4CYP2C9GPR119KCNH2
SCHEMBL1129187 0.84 CYP3A4 (0.61) CYP3A4CYP2C9GPR119KCNH2
SCHEMBL4356654 0.84 CYP3A4 (0.51) CYP3A4CYP2C9GPR119BTK
SCHEMBL4354583 0.84 CYP3A4 (0.60) CYP3A4CYP2C9KCNH2BTK
SCHEMBL4355794 0.82 CYP3A4 (0.57) CYP3A4CYP2C9GPR119BTK
SCHEMBL4350405 0.82 CYP3A4 (0.52) CYP3A4CYP2C9KCNH2BTK
SCHEMBL4328580 0.82 CYP3A4 (0.51) CYP3A4CYP2C9GPR119KCNH2BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009141238-A1 GPR119 RECEPTOR AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-11-26 WO disclosed