SCHEMBL4459796

SCHEMBL4459796

NC1=NC=CC(N)(c2cc(C3CC3)[nH]n2)N1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 0.35
PAK4 O96013 2/20 0.33
PAK1 Q13153 2/20 0.33
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
HCAR3 P49019 1/20 0.33
CCNA2 P20248 1/20 0.30
CDK2 P24941 1/20 0.30
CCNA1 P78396 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4473250 0.76 HCAR2 (0.33) HCAR2HCAR3CCNA2CDK2CCNA1
SCHEMBL4459321 0.75 PDE8B (0.31)
SCHEMBL31268294 0.75 CCNK (0.32)
SCHEMBL31268250 0.75 IGF1R (0.34)
SCHEMBL4472550 0.73 HCAR2 (0.33) HCAR2HCAR3
SCHEMBL31268272 0.73 IGF1R (0.42)
SCHEMBL31268293 0.72 IGF1R (0.34)
SCHEMBL31268258 0.69 AURKA (0.30)
SCHEMBL4454785 0.67
SCHEMBL4473245 0.66 HCAR2 (0.35) HCAR2HCAR3CCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO disclosed