SCHEMBL4468071

SCHEMBL4468071

COC(=O)NC(=O)c1cccc2c1CC(=CCCN1CCC(O)(c3ccc(Cl)cc3)CC1)c1cccnc1O2

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 13/20 0.40
OPRM1 P35372 1/20 0.38
OPRL1 P41146 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CCR1 P32246 3/20 0.38
ADRA1A P35348 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL654064 0.92 DRD2 (0.41) DRD2OPRM1OPRL1CCR1ADRA1A
SCHEMBL654062 0.92 DRD2 (0.41) DRD2OPRM1OPRL1CCR1ADRA1A
SCHEMBL654383 0.90 DRD2 (0.43) DRD2OPRM1CCR1ADRA1A
SCHEMBL654381 0.90 DRD2 (0.43) DRD2OPRM1CCR1ADRA1A
SCHEMBL654870 0.90 DRD2 (0.41) DRD2CCR1ADRA1A
SCHEMBL654872 0.90 DRD2 (0.41) DRD2CCR1ADRA1A
SCHEMBL655038 0.89 DRD2 (0.44) DRD2OPRM1OPRL1CCR1ADRA1A
SCHEMBL655036 0.89 DRD2 (0.44) DRD2OPRM1OPRL1CCR1ADRA1A
SCHEMBL655208 0.89 DRD2 (0.44) DRD2ADRA1A
SCHEMBL655210 0.89 DRD2 (0.44) DRD2ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7541365-B2 Chemokine receptor antagonists and methods of use therefor MILLENNIUM PHARMACEUTICALS, INC. (US) 2009-06-02 US disclosed