SCHEMBL4470692

SCHEMBL4470692

N[C@@H]1[C@H]2CN(c3ccc(F)cc3F)C[C@@H]12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHA2 P29317 1/20 0.47
FLT4 P35916 1/20 0.47
GSK3B P49841 1/20 0.47
RARB P10826 1/20 0.47
TBXAS1 P24557 1/20 0.47
SLC6A3 Q01959 1/20 0.47
ALDH1A1 P00352 5/20 0.43
HTT P42858 3/20 0.43
LMNA P02545 3/20 0.43
KDM4E B2RXH2 2/20 0.43
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
XBP1 P17861 1/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GAA P10253 1/20 0.38
KDM1A O60341 2/20 0.37
KDM1B Q8NB78 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3965681 1.00 EPHA2 (0.47) EPHA2FLT4GSK3BRARBTBXAS1
SCHEMBL4635237 0.80 DPP4 (0.47) EPHA2FLT4GSK3BRARBTBXAS1
SCHEMBL4635925 0.79 DPP4 (0.47) CHRM4DPP4DPP9ADRA1BADRA1D
SCHEMBL13783797 0.78 F2RL1 (0.44) ALDH1A1HTTLMNAKDM4EGAA
SCHEMBL4539952 0.75 ALDH1A1 (0.45) ALDH1A1HTTLMNAKDM4EHPGD
SCHEMBL19262544 0.74 BPTF (0.44)
SCHEMBL6926246 0.74 ALDH1A1 (0.42) ALDH1A1HTTKDM4ECHRM4L3MBTL1
SCHEMBL4321196 0.73 ALDH1A1 (0.48) ALDH1A1HTTLMNAKDM4EPOLB
Hydrochloric Acid SCHEMBL3955678 0.73 DPP4 (0.41) EPHA2FLT4GSK3BRARBTBXAS1
SCHEMBL24018033 0.72 CHRM4 (0.48) EPHA2FLT4GSK3BRARBTBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009090548-A2 3-AZABICYCLO [3.1.0] HEXANE DERIVATIVES AS VANILLOID RECEPTOR LIGANDS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-07-23 WO disclosed