SCHEMBL4471041

SCHEMBL4471041

O=C1COc2ccc(CCc3c[c]ccc3)cc2N1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.58
NR3C2 P08235 3/20 0.56
DRD2 P14416 4/20 0.48
DRD4 P21917 3/20 0.48
DRD3 P35462 2/20 0.48
MMP12 P39900 1/20 0.48
PKM P14618 1/20 0.45
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
HTR1A P08908 5/20 0.44
HTR1D P28221 4/20 0.44
HTR1B P28222 4/20 0.44
SLC6A4 P31645 4/20 0.44
HTR2A P28223 2/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11002313 0.85 PARP1 (0.77) PARP1NR3C2DRD2DRD4DRD3
SCHEMBL4272979 0.84 PARP1 (0.73) PARP1NR3C2DRD2DRD4DRD3
SCHEMBL4263455 0.80 PARP1 (0.60) PARP1NR3C2DRD2DRD4DRD3
SCHEMBL20614334 0.80 MMP12 (0.65) PARP1NR3C2DRD2DRD4DRD3
SCHEMBL7132 0.80 NR3C2 (0.72) PARP1NR3C2DRD2DRD4DRD3
SCHEMBL4257167 0.79 PARP1 (0.70) PARP1NR3C2DRD2DRD4DRD3
SCHEMBL4273023 0.79 PARP1 (0.56) PARP1NR3C2DRD2DRD4DRD3
SCHEMBL4259329 0.79 PARP1 (0.65) PARP1NR3C2DRD2DRD4DRD3
SCHEMBL11006154 0.78 PARP1 (0.70) PARP1NR3C2DRD2DRD4DRD3
SCHEMBL11004751 0.78 PARP1 (0.70) PARP1NR3C2DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009145360-A1 BENZENE OR THIOPHENE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-TECH UENO, LTD. (JP) 2009-12-03 WO disclosed