SCHEMBL4474751

SCHEMBL4474751

O=C(CCNCc1ncc[nH]1)Nc1cccc(NC(=O)CCN2CCC(OC(=O)N(c3ccccc3-c3ccccc3)c3ccccc3-c3ccccc3)CC2)c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 15/20 0.44
ADRB2 P07550 9/20 0.44
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
CCR3 P51677 1/20 0.40
HTR1A P08908 1/20 0.40
HTR7 P34969 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4474750 0.93 CHRM3 (0.41) CHRM3ADRB2DRD2DRD4DRD3
SCHEMBL4478705 0.91 CHRM3 (0.41) CHRM3ADRB2CCR3HTR1AHTR7
SCHEMBL265982 0.90 CHRM3 (0.53) CHRM3ADRB2
SCHEMBL4493379 0.85 CHRM3 (0.47) CHRM3ADRB2NPSR1
SCHEMBL4475320 0.85 CHRM3 (0.49) CHRM3ADRB2NPSR1
SCHEMBL4482057 0.85 CHRM3 (0.48) CHRM3ADRB2
SCHEMBL4478702 0.85 CHRM3 (0.39) CHRM3ADRB2DRD2DRD4DRD3
SCHEMBL4494236 0.84 CHRM3 (0.43) CHRM3ADRB2HTR1AHTR7NPSR1
SCHEMBL265189 0.81 CHRM3 (0.49) CHRM3ADRB2
SCHEMBL4490147 0.80 HTR7 (0.38) CHRM3ADRB2HTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632847-B2 Bronchodilators; treating chronic obstructive pulmonary disease or asthma; long duration of action; reduced side effects, such as dry-mouth and constipation; e.g. biphenyl-2-ylcarbamic acid 1-(2-(3-[3-(4-hydroxybenzylamino)propionylamino]benzoylamino)ethyl)piperidin-4-yl ester THERAVANCE, INC. (US) 2009-12-15 US disclosed