SCHEMBL4478129

SCHEMBL4478129

CCOC(=O)c1cc([N+](=O)[O-])cnc1NOCc1ccccc1.O=c1c(-c2ccccc2)c(O)c2cc([N+](=O)[O-])cnc2n1OCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.39
POLB P06746 2/20 0.39
NFKB1 P19838 3/20 0.38
NFKB2 Q00653 3/20 0.38
RELA Q04206 3/20 0.38
FOS P01100 1/20 0.38
JUN P05412 1/20 0.38
KMT2A Q03164 4/20 0.37
KDM4E B2RXH2 4/20 0.37
MEN1 O00255 3/20 0.37
AR P10275 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TSHR P16473 2/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
CCNA2 P20248 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3517898 0.84 FASN (0.42) MAPTPOLBKMT2AMEN1NPC1
SCHEMBL3514831 0.82 SMN1; SMN2 (0.46) MAPTPOLBKMT2AKDM4EMEN1
SCHEMBL3544652 0.74 KDM4E (0.42) MAPTKMT2AKDM4EMEN1ALDH1A1
SCHEMBL3516064 0.72 MAOB (0.42) MAPTPOLBKMT2AKDM4EMEN1
SCHEMBL3514409 0.72 MAOB (0.47) MAPTPOLBKMT2AKDM4EMEN1
SCHEMBL3517692 0.71 KDM4E (0.47) MAPTKMT2AKDM4EMEN1ALDH1A1
SCHEMBL3519161 0.71 ALDH1A1 (0.38) MAPTKMT2AKDM4EALDH1A1TSHR
SCHEMBL3517053 0.70 MAPK8 (0.39) KMT2AKDM4EALDH1A1TSHRSMN1; SMN2
SCHEMBL3516535 0.70 ALDH1A1 (0.38) MAPTPOLBKMT2AKDM4EMEN1
SCHEMBL3516982 0.69 KDM4E (0.47) MAPTKMT2AKDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044068-A1 1-HYDROXY NAPHTHYRIDINE COMPOUNDS AS ANTI-HIV AGENTS Merck & Co., Inc. (US) 2009-04-08 EP disclosed
WO-2008010964-A1 1-HYDROXY NAPHTHYRIDINE COMPOUNDS AS ANTI-HIV AGENTS MERCK & CO., INC. (US) 2008-01-24 WO disclosed