SCHEMBL4478639

SCHEMBL4478639

O=C(CCN1CCC(OC(=O)N(c2ccccc2-c2ccccc2)c2ccccc2-c2ccccc2)CC1)Nc1cccc(C(=O)NCCNCc2ccco2)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 11/20 0.41
ADRB2 P07550 10/20 0.41
EPHX2 P34913 1/20 0.41
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 1/20 0.39
HTR7 P34969 3/20 0.39
HTR1A P08908 2/20 0.39
HIF1A Q16665 1/20 0.39
EPAS1 Q99814 1/20 0.39
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4478638 0.94 EPHX2 (0.39) CHRM3ADRB2EPHX2TSHRMAPK1
SCHEMBL4494236 0.91 CHRM3 (0.43) CHRM3ADRB2TSHRMAPK1NPC1
SCHEMBL265402 0.91 CHRM3 (0.49) CHRM3ADRB2
SCHEMBL4490821 0.88 CHRM3 (0.43) CHRM3ADRB2EPHX2HTR7HTR1A
SCHEMBL4493225 0.88 CHRM3 (0.46) CHRM3ADRB2EPHX2
SCHEMBL4483296 0.88 CHRM3 (0.45) CHRM3ADRB2
SCHEMBL4474959 0.87 HTR7 (0.39) CHRM3ADRB2EPHX2TSHRMAPK1
SCHEMBL4478705 0.85 CHRM3 (0.41) CHRM3ADRB2EPHX2HTR7HTR1A
SCHEMBL4494233 0.84 CHRM3 (0.41) CHRM3ADRB2TSHRMAPK1NPC1
SCHEMBL4475461 0.82 CHRM3 (0.46) CHRM3ADRB2EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632847-B2 Bronchodilators; treating chronic obstructive pulmonary disease or asthma; long duration of action; reduced side effects, such as dry-mouth and constipation; e.g. biphenyl-2-ylcarbamic acid 1-(2-(3-[3-(4-hydroxybenzylamino)propionylamino]benzoylamino)ethyl)piperidin-4-yl ester THERAVANCE, INC. (US) 2009-12-15 US disclosed