SCHEMBL4479787

SCHEMBL4479787

CC(=O)c1cccc(-c2ccc3c(NC(=O)c4ccccc4)n[nH]c3c2)c1

nearest known ligand 0.73

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 2/20 0.73
FGFR2 P21802 2/20 0.73
FGFR3 P22607 2/20 0.73
HDAC6 Q9UBN7 11/20 0.71
AAK1 Q2M2I8 3/20 0.63
GSK3B P49841 2/20 0.60
CDK7 P50613 2/20 0.58
GSK3A P49840 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4492680 0.89 HDAC6 (0.64) FGFR1FGFR2FGFR3HDAC6AAK1
SCHEMBL4490174 0.89 HDAC6 (0.70) FGFR1FGFR2FGFR3HDAC6AAK1
SCHEMBL4498043 0.89 GSK3B (0.61) FGFR1FGFR2FGFR3HDAC6AAK1
SCHEMBL4494234 0.87 FGFR1 (0.56) FGFR1FGFR2FGFR3HDAC6AAK1
SCHEMBL4506341 0.87 HDAC6 (0.59) FGFR1FGFR2FGFR3HDAC6AAK1
SCHEMBL4486523 0.87 FGFR2 (0.55) FGFR1FGFR2FGFR3HDAC6AAK1
SCHEMBL4489464 0.86 FGFR2 (0.55) FGFR1FGFR2FGFR3HDAC6AAK1
SCHEMBL4484176 0.85 HDAC6 (0.60) FGFR1FGFR2FGFR3HDAC6AAK1
SCHEMBL4498565 0.85 HDAC6 (0.59) FGFR1FGFR2FGFR3HDAC6AAK1
SCHEMBL4502571 0.85 MAPK1 (0.55) FGFR1FGFR2FGFR3HDAC6AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632854-B2 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them PFIZER ITALIA S.R.L. (IT) 2009-12-15 US claimed