SCHEMBL4486523

SCHEMBL4486523

CC(=O)c1cccc(-c2ccc3c(NC(=O)c4c(F)cccc4F)n[nH]c3c2)c1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 4/20 0.55
FGFR3 P22607 4/20 0.55
FGFR1 P11362 3/20 0.55
HDAC6 Q9UBN7 9/20 0.55
AAK1 Q2M2I8 4/20 0.54
GSK3B P49841 3/20 0.53
GSK3A P49840 1/20 0.53
FGFR4 P22455 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4484342 0.93 HDAC6 (0.53) FGFR2FGFR3FGFR1HDAC6AAK1
SCHEMBL4488584 0.93 HDAC6 (0.59) FGFR2FGFR3FGFR1HDAC6GSK3B
SCHEMBL4494234 0.90 FGFR1 (0.56) FGFR2FGFR3FGFR1HDAC6AAK1
SCHEMBL4498043 0.89 GSK3B (0.61) FGFR2FGFR3FGFR1HDAC6AAK1
SCHEMBL4506341 0.88 HDAC6 (0.59) FGFR2FGFR3FGFR1HDAC6AAK1
SCHEMBL4490307 0.87 HDAC6 (0.57) FGFR2FGFR3FGFR1HDAC6AAK1
SCHEMBL4479787 0.87 FGFR1 (0.73) FGFR2FGFR3FGFR1HDAC6AAK1
SCHEMBL4502187 0.87 GSK3B (0.69) FGFR2FGFR3FGFR1HDAC6AAK1
SCHEMBL4480650 0.86 GSK3B (0.54) FGFR2FGFR3FGFR1HDAC6AAK1
SCHEMBL4494537 0.86 FGFR2 (0.52) FGFR2FGFR3FGFR1HDAC6AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632854-B2 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them PFIZER ITALIA S.R.L. (IT) 2009-12-15 US claimed