SCHEMBL4480446

SCHEMBL4480446

Cc1ccc(-c2ccc3c(NC(=O)c4ccccc4F)n[nH]c3c2)cc1C

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 8/20 0.56
HDAC6 Q9UBN7 4/20 0.56
FGFR1 P11362 2/20 0.54
FGFR2 P21802 2/20 0.54
FGFR3 P22607 2/20 0.54
GSK3B P49841 5/20 0.51
CYP1A2 P05177 1/20 0.49
GSK3A P49840 2/20 0.49
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC8 Q9BY41 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4488980 0.89 FGFR4 (0.70) FGFR4HDAC6FGFR1FGFR2FGFR3
SCHEMBL4500056 0.88 HDAC6 (0.55) FGFR4HDAC6FGFR1FGFR2FGFR3
SCHEMBL4495684 0.88 FGFR4 (0.61) FGFR4HDAC6FGFR1FGFR2FGFR3
SCHEMBL4483627 0.88 GSK3B (0.54) FGFR4HDAC6FGFR1FGFR2FGFR3
SCHEMBL4486051 0.88 HDAC6 (0.63) FGFR4HDAC6FGFR1FGFR2FGFR3
SCHEMBL4489919 0.88 HDAC6 (0.54) FGFR4HDAC6FGFR1FGFR2FGFR3
SCHEMBL4482482 0.88 HDAC6 (0.57) FGFR4HDAC6FGFR1FGFR2FGFR3
SCHEMBL4475921 0.86 HDAC6 (0.53) FGFR4HDAC6FGFR1FGFR2FGFR3
SCHEMBL4481006 0.86 HDAC6 (0.60) FGFR4HDAC6FGFR1FGFR2FGFR3
SCHEMBL4488592 0.86 GSK3B (0.66) FGFR4HDAC6FGFR1FGFR2FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632854-B2 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them PFIZER ITALIA S.R.L. (IT) 2009-12-15 US claimed