SCHEMBL4481006

SCHEMBL4481006

CC(=O)c1ccc(-c2ccc3c(NC(=O)c4ccccc4F)n[nH]c3c2)cc1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 10/20 0.60
FGFR1 P11362 1/20 0.58
FGFR2 P21802 1/20 0.58
FGFR3 P22607 1/20 0.58
FGFR4 P22455 5/20 0.54
GSK3B P49841 3/20 0.53
GSK3A P49840 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4494234 0.92 FGFR1 (0.56) HDAC6FGFR1FGFR2FGFR3FGFR4
SCHEMBL4497843 0.88 GSK3B (0.56) HDAC6FGFR1FGFR2FGFR3GSK3B
SCHEMBL4488584 0.88 HDAC6 (0.59) HDAC6FGFR1FGFR2FGFR3GSK3B
SCHEMBL4504535 0.86 FGFR1 (0.54) HDAC6FGFR1FGFR2FGFR3FGFR4
SCHEMBL4496882 0.86 GSK3B (0.62) HDAC6FGFR1FGFR2FGFR3FGFR4
SCHEMBL4480446 0.86 FGFR4 (0.56) HDAC6FGFR1FGFR2FGFR3FGFR4
SCHEMBL4488980 0.86 FGFR4 (0.70) HDAC6FGFR1FGFR2FGFR3FGFR4
SCHEMBL4495684 0.85 FGFR4 (0.61) HDAC6FGFR1FGFR2FGFR3FGFR4
SCHEMBL4488592 0.85 GSK3B (0.66) HDAC6FGFR1FGFR2FGFR3FGFR4
SCHEMBL4502956 0.84 HDAC6 (0.74) HDAC6FGFR1FGFR2FGFR3FGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632854-B2 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them PFIZER ITALIA S.R.L. (IT) 2009-12-15 US claimed