SCHEMBL448148

SCHEMBL448148

COc1cocn1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17394565 0.78
SCHEMBL6959485 0.74
SCHEMBL21966111 0.73
SCHEMBL14031855 0.69 CYP2C19 (0.41)
SCHEMBL14480206 0.69
SCHEMBL14480207 0.69
SCHEMBL17074393 0.69 SCN9A (0.41)
SCHEMBL14031848 0.67 CYP1A2 (0.36)
SCHEMBL1538315 0.66 ALDH1A1 (0.44)
SCHEMBL4164173 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 79 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102911133-B Purification method of (4R,5R)-2- dichloromethyl-4,5- dihydro-5-(4-methylsulfonyl-phenyl)-4-oxazol methanol Shaoxing minsheng pharmaceutical co ltd 2014-07-02 CN claimed
CN-101020666-B Preparation of florfenicol intermediate BAOGUI KE 2011-09-28 CN claimed
CN-101200441-A Preparation of thiamphenicol BAOGUI KE (CN) 2008-06-18 CN claimed
CN-101020666-A Prepn of florfenicol intermediate KE BAOGUI (CN) 2007-08-22 CN claimed
CN-107106558-A Having a2AAminopyrazine compounds with antagonist properties 默沙东公司 2017-08-29 CN disclosed
EP-2997824-A1 NOVEL HERBICIDES Syngenta Participations AG. (CH) 2016-03-23 EP disclosed
CN-105295958-A Liquid crystal aligning agent, liquid crystal alignment film and liquid crystal display element CHI MEI CORP 2016-02-03 CN disclosed
EP-2375898-B1 NOVEL HERBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2015-09-16 EP disclosed
US-8889595-B2 Herbicides SYNGENTA PARTICIPATIONS AG (CH) 2014-11-18 US disclosed
CN-102149675-B Reagents and methods for the synthesis of beta-ketoamide as a precursor to the synthesis of immune adjuvant E6020 EISAI R&D MAN CO LTD 2014-08-20 CN disclosed
CN-102911133-B Purification method of (4R,5R)-2- dichloromethyl-4,5- dihydro-5-(4-methylsulfonyl-phenyl)-4-oxazol methanol Shaoxing minsheng pharmaceutical co ltd 2014-07-02 CN disclosed
CN-103570705-A Substituted N-((1', 3'-azole-4'-yl)-methyl)-4-benzoyl-hexahydropyridine compound and applications thereof INST MEDICINAL BIOTECHNOLOGY 2014-02-12 CN disclosed
US-4956257-A Support with a chemically sensitized silver halide emulsion layer, a hydrophillic colloid layer with a hydrazine compound and a colorless compound with an absorption maxima outside the visible light region FUJI PHOTO FILM CO., LTD. (JP) 1990-09-11 US disclosed
US-4914002-A High contrast image, high sensitivity FUJI PHOTO FILM CO., LTD. (JP) 1990-04-03 US disclosed
EP-0315155-A2 Silver halide photographic material FUJI PHOTO FILM CO., LTD. (JP) 1989-05-10 EP disclosed
EP-0314104-A2 Silver halide photographic materials FUJI PHOTO FILM CO., LTD. (JP) 1989-05-03 EP disclosed
EP-0306019-A2 Silver halide photographic material and method for forming an image FUJI PHOTO FILM CO., LTD. (JP) 1989-03-08 EP disclosed
US-4769316-A Method for restraining the formation of re-reversal negative image in direct positive silver halide photographic materials FUJI PHOTO FILM CO., LTD. (JP) 1988-09-06 US disclosed
US-4607006-A Silver halide photographic light-sensitive material containing non-spectral sensitizing electron donative silver halide adsorptive compound FUJI PHOTO FILM CO., LTD. (JP) 1986-08-19 US disclosed
US-3935010-A IMIDAZOQUINOXALINE DESENSITIZER EASTMAN KODAK COMPANY (US) 1976-01-27 US disclosed