Bp-14979

Bp-14979

SCHEMBL4482277

COCCC(=O)NC1CCC(CCN2CCN(c3cccc(C#N)c3)CC2)CC1

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 15/20 0.63
DRD3 P35462 15/20 0.63
HTR2A P28223 11/20 0.63
HTR1A P08908 4/20 0.63
DRD4 P21917 4/20 0.63
HTR2B P41595 4/20 0.63
HTR2C P28335 3/20 0.63
DRD1 P21728 1/20 0.63
CHRM4 P08173 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bp-14979 SCHEMBL24005999 1.00 DRD2 (0.63) DRD2DRD3HTR2AHTR1ADRD4
Bp-14979 SCHEMBL29730885 1.00 DRD2 (0.63) DRD2DRD3HTR2AHTR1ADRD4
Bp-14979 SCHEMBL13630506 1.00 DRD2 (0.63) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL13630394 0.95 DRD2 (0.57) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL4490376 0.95 DRD2 (0.57) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL25535948 0.91 DRD2 (0.66) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL13629925 0.91 DRD2 (0.60) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL4483671 0.91 DRD2 (0.60) DRD2DRD3HTR2AHTR1ADRD4
Bp-14979 SCHEMBL17220515 0.90 DRD2 (0.55) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL13630505 0.88 DRD2 (0.64) DRD2DRD3HTR2ACHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12582648-B2 Method for treating central nervous system disorders using dopamine D3 partial agonists BIOPROJET PHARMA (FR) 2026-03-24 US claimed
US-20230165852-A1 METHOD FOR TREATING CENTRAL NERVOUS SYSTEM DISORDERS USING DOPAMINE D3 PARTIAL AGONISTS BIOPROJET PHARMA (FR) 2023-06-01 US claimed
EP-4146214-A1 USE OF DOPAMINE D3 PARTIAL AGONISTS FOR TREATING CENTRAL NERVOUS SYSTEM DISORDERS BIOPROJET Pharma (FR) 2023-03-15 EP claimed
CN-115715195-A Use of partial dopamine D3 agonists for the treatment of central nervous system disorders 生物计划制药公司 2023-02-24 CN claimed
EP-3906927-B1 USE OF DOPAMINE D3 PARTIAL AGONISTS FOR TREATING CENTRAL NERVOUS SYSTEM DISORDERS BIOPROJET PHARMA (FR) 2022-05-25 EP claimed
EP-3906927-A1 USE OF DOPAMINE D3 PARTIAL AGONISTS FOR TREATING CENTRAL NERVOUS SYSTEM DISORDERS BIOPROJET Pharma (FR) 2021-11-10 EP claimed
EP-2038268-B1 CARBONYLATED (AZA)CYCLOHEXANES AS DOPAMINE D3 RECEPTOR LIGANDS BIOPROJET SOC CIV (FR) 2015-11-04 EP claimed
US-8802678-B2 Carbonylated (aza) cyclohexanes as dopamine D3 receptor ligands BIOPROJET (FR) 2014-08-12 US claimed
US-20090286801-A1 CARBONYLATED (AZA) CYCLOHEXANES AS DOPAMINE D3 RECEPTOR LIGANDS BIOPROJET (FR) 2009-11-19 US claimed
US-12582648-B2 Method for treating central nervous system disorders using dopamine D3 partial agonists BIOPROJET PHARMA (FR) 2026-03-24 US disclosed
US-20230165852-A1 METHOD FOR TREATING CENTRAL NERVOUS SYSTEM DISORDERS USING DOPAMINE D3 PARTIAL AGONISTS BIOPROJET PHARMA (FR) 2023-06-01 US disclosed
EP-4146214-A1 USE OF DOPAMINE D3 PARTIAL AGONISTS FOR TREATING CENTRAL NERVOUS SYSTEM DISORDERS BIOPROJET Pharma (FR) 2023-03-15 EP disclosed
CN-115715195-A Use of partial dopamine D3 agonists for the treatment of central nervous system disorders 生物计划制药公司 2023-02-24 CN disclosed
EP-3906927-B1 USE OF DOPAMINE D3 PARTIAL AGONISTS FOR TREATING CENTRAL NERVOUS SYSTEM DISORDERS BIOPROJET PHARMA (FR) 2022-05-25 EP disclosed
WO-2021224235-A1 USE OF DOPAMINE D3 PARTIAL AGONISTS FOR TREATING CENTRAL NERVOUS SYSTEM DISORDERS BIOPROJET PHARMA (FR) 2021-11-11 WO disclosed
EP-3906927-A1 USE OF DOPAMINE D3 PARTIAL AGONISTS FOR TREATING CENTRAL NERVOUS SYSTEM DISORDERS BIOPROJET Pharma (FR) 2021-11-10 EP disclosed
EP-3906927-A1 USE OF DOPAMINE D3 PARTIAL AGONISTS FOR TREATING CENTRAL NERVOUS SYSTEM DISORDERS BIOPROJET Pharma (FR) 2021-11-10 EP disclosed
EP-2038268-B1 CARBONYLATED (AZA)CYCLOHEXANES AS DOPAMINE D3 RECEPTOR LIGANDS BIOPROJET SOC CIV (FR) 2015-11-04 EP disclosed
US-8802678-B2 Carbonylated (aza) cyclohexanes as dopamine D3 receptor ligands BIOPROJET (FR) 2014-08-12 US disclosed
US-20090286801-A1 CARBONYLATED (AZA) CYCLOHEXANES AS DOPAMINE D3 RECEPTOR LIGANDS BIOPROJET (FR) 2009-11-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090286801-A1 CARBONYLATED (AZA) CYCLOHEXANES AS DOPAMINE D3 RECEPTOR LIGANDS DRD3, TACR2, TACR1 DRD2 4/4885DRD3 1/4885HTR2A 225/4885
US-12582648-B2 Method for treating central nervous system disorders using dopamine D3 partial agonists DRD3, DRD2, DRD1 DRD2 2/4885DRD3 1/4885HTR2A 209/4885
US-20230165852-A1 METHOD FOR TREATING CENTRAL NERVOUS SYSTEM DISORDERS USING DOPAMINE D3 PARTIAL AGONISTS DRD3, DRD2, DRD1 DRD2 2/4885DRD3 1/4885HTR2A 71/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.