SCHEMBL4482463

SCHEMBL4482463

Oc1ccc(-n2ccnn2)cc1-n1ccnn1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 17/20 0.54
KEAP1 Q14145 1/20 0.49
CYP19A1 P11511 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4564455 0.81 NOTUM (0.58) NOTUMKEAP1CYP19A1
SCHEMBL13735664 0.81 NOTUM (0.58) NOTUMKEAP1CYP19A1
SCHEMBL2359098 0.79 NOTUM (0.54) NOTUMKEAP1CYP19A1
SCHEMBL5612825 0.77 NOTUM (0.53) NOTUMKEAP1CYP19A1
SCHEMBL22325390 0.77 NOTUM (0.53) NOTUMKEAP1CYP19A1
SCHEMBL4457296 0.77 NOTUM (0.49) NOTUMKEAP1
SCHEMBL10447781 0.76 NOTUM (0.78) NOTUMKEAP1CYP19A1
SCHEMBL1696198 0.76 NOTUM (0.47) NOTUMKEAP1
SCHEMBL17422567 0.76 NOTUM (0.51) NOTUMKEAP1
SCHEMBL5602626 0.76 NOTUM (0.47) NOTUMKEAP1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2034996-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY Synta Pharmaceuticals Corporation (US) 2009-03-18 EP claimed
WO-2007139955-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2007-12-06 WO claimed
EP-2034996-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY Synta Pharmaceuticals Corporation (US) 2009-03-18 EP disclosed
WO-2007139955-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2007-12-06 WO disclosed