Mometasone Furoate

Mometasone Furoate

SCHEMBL4484

C[C@@H]1C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)C3(Cl)[C@@H](O)C[C@]2(C)[C@@]1(OC(=O)c1ccco1)C(=O)CCl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

NR3C1

The experimentally established mechanism targets of Mometasone Furoate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 known ✓ P04150 5/20 1.00
CYP3A4 P08684 7/20 1.00
LMNA P02545 5/20 1.00
ABCB11 O95342 4/20 1.00
PGR P06401 4/20 1.00
AR P10275 3/20 1.00
ADORA3 P0DMS8 2/20 1.00
CYP2D6 P10635 2/20 1.00
CYP2C9 P11712 2/20 1.00
PTGS1 P23219 2/20 1.00
CYP1A2 P05177 1/20 1.00
CYP2C19 P33261 1/20 1.00
SLCO1B3 Q9NPD5 1/20 1.00
SLCO1B1 Q9Y6L6 1/20 1.00
USP2 O75604 4/20 0.64
HIF1A Q16665 3/20 0.64
CNR1 P21554 2/20 0.64
CHRM1 P11229 1/20 0.64
TBXA2R P21731 1/20 0.64
MAPT P10636 3/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mometasone Furoate SCHEMBL4568 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL8430908 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL12996648 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL4896227 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL8826257 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL7436523 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL25382496 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL2594997 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL13026146 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL600107 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 26692 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137657-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US claimed
US-20260137656-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US claimed
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
US-20260130899-A1 METHOD OF TREATMENT FOR PREVENTION OF GLUCOCORTICOID TOXICITY AND/OR ENHANCEMENT OF MUSCLE REGENERATION VIA NEUTROPHIL ELASTASE INHIBITION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2026-05-14 US claimed
US-20260125686-A1 COMPOSITIONS AND METHODS FOR MODULATION OF CFTR CYSTIC FIBROSIS FOUND (US) 2026-05-07 US claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-4736841-A1 A MUCOADHESIVE LAYER FOR BUCCAL ADMINISTRATION OF AN ACTIVE PHARMACEUTICAL INGREDIENT IQ medical GmbH (DE) 2026-05-06 EP claimed
EP-4735431-A2 MK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. (US) 2026-05-06 EP claimed
US-12616803-B2 Apparatus for dispensing inhalant medicament METOPI PHARMACEUTICALS, INC. (US) 2026-05-05 US claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
CN-1133004-A Method for regulating substances ASTRA AB (SE) 1996-10-09 CN claimed
WO-1996024359-A1 NOVEL PHARMACEUTICAL FORMULATION ASTRA AKTIEBOLAG (SE) 1996-08-15 WO claimed
WO-1996024355-A1 NOVEL PHARMACEUTICAL COMBINATION ASTRA AKTIEBOLAG (SE) 1996-08-15 WO claimed
EP-0721348-A1 MONOGLYCERIDE/LACTATE ESTER PERMEATION ENHANCER ALZA CORPORATION (US) 1996-07-17 EP claimed
WO-1996019198-A1 AEROSOL DRUG FORMULATIONS ASTRA AKTIEBOLAG (SE) 1996-06-27 WO claimed
EP-0292893-B2 Steroid lotion SCHERING CORP (US) 1995-11-29 EP claimed
US-5407663-A Swishing solution in mouth, expectorating EISEN DRORE (US) 1995-04-18 US claimed
WO-1995009006-A1 MONOGLYCERIDE/LACTATE ESTER PERMEATION ENHANCER ALZA CORPORATION (US) 1995-04-06 WO claimed
EP-0548114-B1 MOMETASONE FUROATE MONOHYDRATE, PROCESS FOR MAKING SAME AND PHARMACEUTICAL COMPOSITIONS SCHERING CORP (US) 1994-11-02 EP claimed
EP-0262681-B1 ANTI-INFLAMMATORY CREAM COMPOSITION SCHERING CORPORATION (US) 1991-04-24 EP claimed