Mometasone Furoate

Mometasone Furoate

SCHEMBL4568

C[C@@H]1C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(Cl)[C@@H](O)C[C@]2(C)[C@@]1(OC(=O)c1ccco1)C(=O)CCl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

NR3C1

The experimentally established mechanism targets of Mometasone Furoate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 known ✓ P04150 5/20 1.00
CYP3A4 P08684 7/20 1.00
LMNA P02545 5/20 1.00
ABCB11 O95342 4/20 1.00
PGR P06401 4/20 1.00
AR P10275 3/20 1.00
ADORA3 P0DMS8 2/20 1.00
CYP2D6 P10635 2/20 1.00
CYP2C9 P11712 2/20 1.00
PTGS1 P23219 2/20 1.00
CYP1A2 P05177 1/20 1.00
CYP2C19 P33261 1/20 1.00
SLCO1B3 Q9NPD5 1/20 1.00
SLCO1B1 Q9Y6L6 1/20 1.00
USP2 O75604 4/20 0.64
HIF1A Q16665 3/20 0.64
CNR1 P21554 2/20 0.64
CHRM1 P11229 1/20 0.64
TBXA2R P21731 1/20 0.64
MAPT P10636 3/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mometasone Furoate SCHEMBL8430908 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL12996648 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL4896227 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL8826257 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL7436523 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL25382496 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL2594997 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL13026146 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL600107 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR
Mometasone Furoate SCHEMBL4484 1.00 CYP3A4 (1.00) CYP3A4NR3C1LMNAABCB11PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 29009 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026104312-A1 STABLE MOMETASONE FUROATE COMPOSITIONS LTS LOHMANN THERAPIE-SYSTEME AG (DE) 2026-05-21 WO claimed
EP-4744657-A1 THERAPEUTIC AGENT FOR HUMAN GRAFT VERSUS HOST DISEASE AND COMBINATION THEREOF National University Corporation Okayama University (JP) 2026-05-20 EP claimed
CN-122057085-A External auditory canal degradable and self-adaptive drug stent with combined drug release in segmented mode and preparation method thereof 上海交通大学医学院附属瑞金医院 2026-05-19 CN claimed
CN-122031290-A Percutaneous permeation promoting system and preparation method and application thereof 北京工商大学 2026-05-15 CN claimed
US-20260130899-A1 METHOD OF TREATMENT FOR PREVENTION OF GLUCOCORTICOID TOXICITY AND/OR ENHANCEMENT OF MUSCLE REGENERATION VIA NEUTROPHIL ELASTASE INHIBITION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2026-05-14 US claimed
EP-4739295-A1 AN INHALABLE FORMULATION OF FLUTICASONE PROPIONATE AND ALBUTEROL SULFATE FOR THE TREATMENT OF ASTHMA Norton (Waterford) Limited (IE) 2026-05-13 EP claimed
EP-4739294-A1 AN INHALABLE FORMULATION OF FLUTICASONE PROPIONATE AND ALBUTEROL SULFATE FOR THE TREATMENT OF ASTHMA Norton (Waterford) Limited (IE) 2026-05-13 EP claimed
CN-122005510-A Momordant mometasone furoate dry powder inhalant without carrier and preparation method thereof 江苏德迈药业有限公司 2026-05-12 CN claimed
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES TRAILHEAD BIOSYSTEMS INC (US) 2026-05-07 US claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
WO-1991007169-A1 GLYCERYL ACETATE OINTMENT VEHICLES DOW GORDON JAY (US) 1991-05-30 WO claimed
EP-0262681-B1 ANTI-INFLAMMATORY CREAM COMPOSITION SCHERING CORPORATION (US) 1991-04-24 EP claimed
EP-0362270-A1 STEROID LOTION. SCHERING CORP (US) 1990-04-11 EP claimed
EP-0318522-A1 ANTI-INFLAMMATORY CREAM COMPOSITION SCHERING CORPORATION (US) 1989-06-07 EP claimed
US-4808610-A STABILITY, PREGNADIENE COMPOUND SCHERING CORPORATION (US) 1989-02-28 US claimed
WO-1988009174-A1 STEROID LOTION SCHERING CORPORATION (US) 1988-12-01 WO claimed
EP-0292893-A1 Steroid lotion SCHERING CORPORATION (US) 1988-11-30 EP claimed
US-4775529-A ANTIINFLAMMATORY, VASOCONSTRICTION; PROPYLENE GLYCOL; ISOPROPANOL AND THICKENER; SKIN DISORDERS SCHERING CORPORATION (US) 1988-10-04 US claimed
WO-1988002257-A1 ANTI-INFLAMMATORY CREAM COMPOSITION SCHERING CORPORATION (US) 1988-04-07 WO claimed
EP-0262681-A1 Anti-inflammatory cream composition SCHERING CORPORATION (US) 1988-04-06 EP claimed