SCHEMBL4484583

SCHEMBL4484583

COCCNS(=O)(=O)c1ccc(Nc2nccc(-c3cnc4n3CCC4)n2)cc1

nearest known ligand 0.68

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 16/20 0.68
CDK4 P11802 6/20 0.68
CDK1 P06493 3/20 0.58
SYK P43405 1/20 0.46
IKBKB O14920 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4818566 0.81 CDK2 (1.00) CDK2CDK4CDK1
SCHEMBL5108640 0.80 CDK2 (0.81) CDK2CDK4CDK1
SCHEMBL5092316 0.80 CDK2 (1.00) CDK2CDK4CDK1
SCHEMBL5095501 0.80 CDK2 (0.80) CDK2CDK4CDK1
SCHEMBL5105389 0.80 CDK2 (0.72) CDK2CDK4CDK1SYKIKBKB
SCHEMBL23752538 0.79 CDK2 (1.00) CDK2CDK4CDK1
SCHEMBL5098635 0.79 CDK2 (0.79) CDK2CDK4CDK1
SCHEMBL6410272 0.78 CDK2 (0.87) CDK2CDK4CDK1
SCHEMBL6244692 0.78 CDK2 (0.78) CDK2CDK4CDK1IKBKB
SCHEMBL27584963 0.78 CDK2 (1.00) CDK2CDK4CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7579344-B2 Pyrimidine derivatives possessing cell-cycle inhibitors activity ASTRAZENECA AB (SE) 2009-08-25 US disclosed