SCHEMBL4485380

SCHEMBL4485380

CC(C)(C)OC(=O)N1CC2C(C1)C2(C#N)c1ccc(-c2c(F)cc(N3C[C@H](Cn4ccnn4)OC3=O)cc2F)cn1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOA P21397 17/20 0.53
CYP3A4 P08684 3/20 0.47
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
KCNH2 Q12809 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13711500 1.00 MAOA (0.53) MAOACYP3A4CYP2D6CYP2C9KCNH2
SCHEMBL13711597 0.93 MAOA (0.63) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL3368491 0.93 MAOA (0.63) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL3368907 0.92 MAOA (0.47) MAOACYP3A4CYP2D6CYP2C9KCNH2
SCHEMBL3366657 0.91 MAOA (0.47) MAOACYP3A4CYP2C9KCNH2
SCHEMBL3368742 0.91 MAOA (0.47) MAOACYP3A4CYP2D6CYP2C9KCNH2
SCHEMBL3368070 0.91 MAOA (0.49) MAOACYP3A4CYP2D6CYP2C9KCNH2
SCHEMBL13711602 0.91 MAOA (0.49) MAOACYP3A4CYP2D6CYP2C9KCNH2
SCHEMBL13711581 0.90 MAOA (0.49) MAOACYP3A4CYP2D6CYP2C9KCNH2
SCHEMBL3367228 0.90 MAOA (0.49) MAOACYP3A4CYP2D6CYP2C9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582659-B2 Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof MERCK & CO., INC. (US) 2009-09-01 US disclosed
US-7462633-B2 Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof MERCK & CO., INC. (US) 2008-12-09 US disclosed