SCHEMBL4489942

SCHEMBL4489942

CCCCC(=O)Nc1n[nH]c2cc(-c3cccc(Cl)c3)ccc12

nearest known ligand 0.79

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 6/20 0.79
HDAC2 Q92769 6/20 0.79
HDAC8 Q9BY41 6/20 0.79
GSK3B P49841 13/20 0.74
CYP1A2 P05177 2/20 0.64
HDAC6 Q9UBN7 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4499076 0.95 GSK3B (0.83) HDAC1HDAC2HDAC8GSK3BCYP1A2
SCHEMBL4500438 0.87 GSK3B (0.74) HDAC1HDAC2HDAC8GSK3BCYP1A2
SCHEMBL4497459 0.86 GSK3B (0.69) HDAC1HDAC2HDAC8GSK3BCYP1A2
SCHEMBL4503159 0.86 GSK3B (0.70) HDAC1HDAC2HDAC8GSK3BCYP1A2
SCHEMBL1461654 0.85 GSK3B (1.00) GSK3BCYP1A2
SCHEMBL4483697 0.85 HDAC1 (0.69) HDAC1HDAC2HDAC8GSK3BCYP1A2
SCHEMBL1461243 0.84 GSK3B (0.84) HDAC1HDAC2HDAC8GSK3BCYP1A2
SCHEMBL4496059 0.84 GSK3B (0.65) HDAC1HDAC2HDAC8GSK3BCYP1A2
SCHEMBL4493121 0.83 GSK3B (1.00) HDAC1HDAC2HDAC8GSK3BCYP1A2
SCHEMBL31060453 0.83 GSK3B (1.00) HDAC1HDAC2HDAC8GSK3BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632854-B2 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them PFIZER ITALIA S.R.L. (IT) 2009-12-15 US claimed