SCHEMBL449056

SCHEMBL449056

COc1ccc(OC)c(S(=O)(=O)N(C)Cc2nc3ccccc3c(=O)n2-c2ccc(C)cc2C)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
L3MBTL1 Q9Y468 1/20 0.47
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HSD17B10 Q99714 1/20 0.45
HPGD P15428 1/20 0.45
MAPK1 P28482 1/20 0.45
USP2 O75604 1/20 0.44
NPSR1 Q6W5P4 2/20 0.44
PDE10A Q9Y233 1/20 0.44
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
GAA P10253 2/20 0.43
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL448162 0.91 ALDH1A1 (0.48) ALDH1A1L3MBTL1MAPTKDM4ESMN1; SMN2
SCHEMBL449986 0.90 ALDH1A1 (0.53) ALDH1A1L3MBTL1MAPTKDM4ESMN1; SMN2
SCHEMBL454849 0.88 ALDH1A1 (0.53) ALDH1A1L3MBTL1MAPTKDM4ESMN1; SMN2
SCHEMBL448160 0.86 ALDH1A1 (0.51) ALDH1A1L3MBTL1MAPTKDM4ESMN1; SMN2
SCHEMBL451091 0.86 ALDH1A1 (0.51) ALDH1A1L3MBTL1MAPTKDM4ESMN1; SMN2
SCHEMBL453808 0.86 ALDH1A1 (0.56) ALDH1A1L3MBTL1MAPTKDM4ESMN1; SMN2
SCHEMBL450403 0.86 ALDH1A1 (0.56) ALDH1A1L3MBTL1MAPTKDM4ESMN1; SMN2
SCHEMBL449985 0.84 ALDH1A1 (0.54) ALDH1A1L3MBTL1MAPTKDM4ESMN1; SMN2
SCHEMBL450535 0.84 ALDH1A1 (0.48) ALDH1A1MAPTKDM4ESMN1; SMN2HPGD
SCHEMBL450437 0.83 ALDH1A1 (0.53) ALDH1A1L3MBTL1MAPTKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 58 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8748440-B2 Quinazolinone modulators of nuclear receptors EXELIXIS, INC. (US) 2014-06-10 US claimed
US-20120064025-A1 Quinazolinone Modulators Of Nuclear Receptors EXELIXIS, INC. (US) 2012-03-15 US claimed
EP-1521746-B1 QUINAZOLINONE MODULATORS OF NUCLEAR RECEPTORS X CEPTOR THERAPEUTICS INC (US) 2011-04-27 EP claimed
US-20080070864-A1 Quinazolinone Modulators Of Nuclear Receptors X-CEPTOR THERAPEUTICS, INC. (US) 2008-03-20 US claimed
US-20240040853-A1 DISPLAY PANELS, MANUFACTURING METHODS THEREOF, AND DISPLAY DEVICES TCL CHINA STAR OPTOELECTRONICS TECHNOLOGY CO., LTD. (CN) 2024-02-01 US disclosed
EP-4312481-A1 DISPLAY PANELS, MANUFACTURING METHODS THEREOF, AND DISPLAY DEVICES TCL CHINA STAR OPTOELECTRONICS TECHNOLOGY CO., LTD. (CN) 2024-01-31 EP disclosed
US-10665812-B2 Organic EL display panel and method for producing organic EL display panel JOLED INC. (JP) 2020-05-26 US disclosed
US-10263046-B2 Organic EL display panel and method of manufacturing organic EL display panel JOLED INC. (JP) 2019-04-16 US disclosed
US-20180090546-A1 ORGANIC EL DISPLAY PANEL AND METHOD OF MANUFACTURING ORGANIC EL DISPLAY PANEL MAGNOLIA BLUE CORPORATION (JP) 2018-03-29 US disclosed
US-9490444-B2 Organic light-emitting element with regulation insulating layer and two-component electron transport layer and method of making JOLED INC. (JP) 2016-11-08 US disclosed
US-9490445-B2 Organic el element, organic el panel, organic el light-emitting apparatus, organic el display apparatus, and method of manufacturing organic el element JOLED INC. (JP) 2016-11-08 US disclosed
US-9324964-B2 Organic light-emitting element with hole injection layer having concave portion JOLED INC. (JP) 2016-04-26 US disclosed
US-20130126840-A1 ORGANIC EL ELEMENT, ORGANIC EL PANEL, ORGANIC EL LIGHT-EMITTING APPARATUS, ORGANIC EL DISPLAY APPARATUS, AND METHOD OF MANUFACTURING ORGANIC EL ELEMENT PANASONIC CORPORATION (JP) 2013-05-23 US disclosed
US-20130105780-A1 METHOD FOR PRODUCING ORGANIC EL ELEMENT, DISPLAY DEVICE, LIGHT-EMITTING APPARATUS, AND ULTRAVIOLET IRRADIATION DEVICE PANASONIC CORPORATION (JP) 2013-05-02 US disclosed
US-20130056719-A1 ORGANIC EL DISPLAY PANEL AND ORGANIC EL DISPLAY APPARATUS PANASONIC CORPORATION (JP) 2013-03-07 US disclosed
US-20120132934-A1 ORGANIC EL ELEMENT, DISPLAY APPARATUS, AND LIGHT-EMITTING APPARATUS PANASONIC CORPORATION (JP) 2012-05-31 US disclosed
US-20120061656-A1 ORGANIC EL ELEMENT PANASONIC CORPORATION (JP) 2012-03-15 US disclosed
US-20120064025-A1 Quinazolinone Modulators Of Nuclear Receptors EXELIXIS, INC. (US) 2012-03-15 US disclosed
EP-1521746-B1 QUINAZOLINONE MODULATORS OF NUCLEAR RECEPTORS X CEPTOR THERAPEUTICS INC (US) 2011-04-27 EP disclosed
US-20080070864-A1 Quinazolinone Modulators Of Nuclear Receptors X-CEPTOR THERAPEUTICS, INC. (US) 2008-03-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120064025-A1 Quinazolinone Modulators Of Nuclear Receptors NR1H4, NR1H2, NR1H3 ALDH1A1 3161/4885L3MBTL1 4767/4885MAPT 4075/4885
US-20080070864-A1 Quinazolinone Modulators Of Nuclear Receptors NR1H4, NR1H2, NR1H3 ALDH1A1 3161/4885L3MBTL1 4767/4885MAPT 4075/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.