SCHEMBL4491749

SCHEMBL4491749

COc1ccc(-c2ccc3c(NC(=O)CC4CCCC4)n[nH]c3c2)cc1

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 7/20 0.64
HDAC2 Q92769 7/20 0.64
HDAC8 Q9BY41 7/20 0.64
HDAC6 Q9UBN7 1/20 0.59
AAK1 Q2M2I8 1/20 0.56
GSK3B P49841 9/20 0.55
EPHX2 P34913 1/20 0.54
FGFR4 P22455 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4483758 0.91 HDAC1 (0.67) HDAC1HDAC2HDAC8HDAC6AAK1
SCHEMBL4505755 0.90 HDAC1 (0.68) HDAC1HDAC2HDAC8HDAC6GSK3B
SCHEMBL4494068 0.89 HDAC1 (0.54) HDAC1HDAC2HDAC8HDAC6AAK1
SCHEMBL4498522 0.89 HDAC1 (0.55) HDAC1HDAC2HDAC8HDAC6AAK1
SCHEMBL4486080 0.89 GSK3B (0.66) AAK1GSK3B
SCHEMBL4480696 0.87 AAK1 (0.57) AAK1GSK3B
SCHEMBL4483041 0.86 GSK3B (0.67) AAK1GSK3B
SCHEMBL4503278 0.86 GSK3B (0.70) AAK1GSK3B
SCHEMBL4485536 0.85 HDAC6 (0.58) HDAC6AAK1GSK3BFGFR4
SCHEMBL4486782 0.85 HDAC1 (0.68) HDAC1HDAC2HDAC8HDAC6AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632854-B2 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them PFIZER ITALIA S.R.L. (IT) 2009-12-15 US claimed