SCHEMBL4510951

SCHEMBL4510951

Cc1csc2c1c(O)c(C(=O)O)c(=O)n2C

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 6/20 0.51
ERCC5 P28715 4/20 0.51
LDHA P00338 3/20 0.38
LDHB P07195 3/20 0.38
ADORA2B P29275 7/20 0.35
ERCC1 P07992 1/20 0.35
ERCC4 Q92889 1/20 0.35
POLB P06746 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33
ALB P02768 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4517627 0.82 ALDH1A1 (0.51) FEN1ERCC5ADORA2BPOLBTDP1
SCHEMBL15154655 0.82 MEN1 (0.48) FEN1ERCC5
SCHEMBL4509473 0.80 KMT2A (0.57) FEN1ERCC5ADORA2BPOLB
SCHEMBL4510344 0.79 KMT2A (0.56) FEN1ERCC5ADORA2BPOLB
SCHEMBL4506552 0.79 KMT2A (0.56) FEN1ERCC5ADORA2BPOLB
SCHEMBL4507747 0.79 KMT2A (0.56) FEN1ERCC5ADORA2BPOLB
SCHEMBL4496687 0.79 KMT2A (0.56) FEN1ERCC5ADORA2BPOLB
SCHEMBL5236265 0.79 KMT2A (0.56) FEN1ERCC5ADORA2BPOLB
SCHEMBL4506695 0.77 MEN1 (0.42) FEN1ERCC5ADORA2B
SCHEMBL4494251 0.77 MEN1 (0.48) FEN1ERCC5L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1980937-B Thienopyridone carboxamides and their medical use ACTIVE BIOTECH AB 2011-08-10 CN disclosed
US-7553849-B2 Compounds ACTIVE BIOTECH AB (SE) 2009-06-30 US disclosed
EP-1776369-B1 THIENOPYRIDONE CARBOXAMIDES AND THEIR MEDICAL USE ACTIVE BIOTECH AB (SE) 2007-10-10 EP disclosed
CN-1980937-A Thienopyridone carboxamides and their medical use ACTIVE BIOTECH AB (SE) 2007-06-13 CN disclosed
US-20060004038-A1 Novel compounds ACTIVE BIOTECH AB (SE) 2006-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060004038-A1 Novel compounds REL, CLIC4, C5 FEN1 3426/4885ERCC5 1570/4885LDHA 4659/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.