SCHEMBL4515159

SCHEMBL4515159

O=C(NCc1ccc(F)cc1)c1sc2ncccc2c1-c1ccc(F)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.51
MAPT P10636 3/20 0.50
TP53 P04637 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
LMNA P02545 1/20 0.48
CYP1A2 P05177 1/20 0.48
CHRM4 P08173 1/20 0.48
CYP2D6 P10635 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13605653 0.95 MAPT (0.58) KMT2AMAPTTP53RXFP1LMNA
SCHEMBL8239164 0.87 EGLN1 (0.44) MAPTTP53
SCHEMBL13605661 0.84 TP53 (0.45) KMT2AMAPTTP53CYP1A2
SCHEMBL4518456 0.83 MAPT (0.43) MAPT
SCHEMBL8241900 0.83 ADORA2A (0.56) KMT2AMAPTLMNA
SCHEMBL4524608 0.82 KAT2B (0.42) MAPTTP53LMNA
SCHEMBL4533208 0.81 KDM4E (0.49)
Hydrochloric Acid SCHEMBL4520231 0.80 KDM4E (0.48)
SCHEMBL8239980 0.80 IKBKB (0.43)
SCHEMBL27724629 0.80 TP53 (0.55) KMT2AMAPTTP53LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090326001-A1 THIENOPYRIDINE DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS RICHTER GEDEON NYRT. (HU) 2009-12-31 US claimed
EP-4584250-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS Biohaven Therapeutics Ltd. (VG) 2025-07-16 EP disclosed
WO-2024054811-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS BIOHAVEN THERAPEUTICS LTD. (VG) 2024-03-14 WO disclosed
US-20090326001-A1 THIENOPYRIDINE DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS RICHTER GEDEON NYRT. (HU) 2009-12-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090326001-A1 THIENOPYRIDINE DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS GRM5, GRM1, GRIK5 KMT2A 2966/4885MAPT 1718/4885TP53 4881/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.