Triaziquone

Triaziquone

SCHEMBL451592

CCS(=O)(=O)O.O=C1C=C(N2CC2)C(=O)C(N2CC2)=C1N1CC1

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

FGFR1FGFR2FGFR3FGFR4FLT1FLT4KDRPDGFRAPDGFRB

The experimentally established mechanism targets of Triaziquone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.40
HTT P42858 2/20 0.40
TP53 P04637 1/20 0.40
STAT3 P40763 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DNMT1 P26358 1/20 0.39
NSD2 O96028 3/20 0.35
TTR P02766 1/20 0.35
APAF1 O14727 2/20 0.33
TDP2 O95551 2/20 0.33
HKDC1 Q2TB90 2/20 0.33
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
HIF1A Q16665 1/20 0.31
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triaziquone SCHEMBL17874437 0.89 HTT (0.42) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL11350903 0.89 HTT (0.42) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL9791390 0.87 DNMT1 (0.42) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL21358774 0.87 MAPT (0.43) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL7783197 0.87 MAPT (0.46) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL33439 0.86 HTT (0.42) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL8965684 0.85 HTT (0.39) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL149876 0.83 MAPT (0.46) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL6225692 0.83 TP53 (0.38) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL6000230 0.83 DNMT1 (0.47) MAPTHTTTP53STAT3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114634886-A Multifunctional microbial agent capable of degrading various halogenated organic pollutants simultaneously 河南科技大学 2022-06-17 CN claimed
CN-114394680-A Application of microbial agent in degradation of various halogenated organic pollutants 河南科技大学 2022-04-26 CN claimed
CN-110038635-B Acetylene dimerization aqueous phase catalyst and application thereof 石河子大学 2022-02-11 CN claimed
CN-111676147-A Method for enriching and separating dechlorinating tetrachloroethylene bacteria and application 中山大学 2020-09-18 CN claimed
CN-111569152-A Biological valve with anticoagulation and calcification resistance and preparation method thereof 四川大学 2020-08-25 CN claimed
CN-110038635-A A kind of acetylene dimer aqueous phase catalyst and its application 石河子大学 2019-07-23 CN claimed
EP-2774630-B1 METHOD FOR PREPARING EDGE-RIGIDIZED ARTIFICIAL BIOLOGICAL VALVE SHANGHAI MICROPORT CARDIOFLOW MEDTECH CO LTD (CN) 2017-07-05 EP claimed
EP-2774630-A1 METHOD FOR PREPARING EDGE-RIGIDIZED ARTIFICIAL BIOLOGICAL VALVE Shanghai MicroPort Medical (Group) Co., Ltd. (CN) 2014-09-10 EP claimed
CN-118345123-A Method for producing chemicals by artificial light driven microbial flora in low carbon 南京工业大学 2024-07-16 CN disclosed
CN-118324293-A Carbon-based adsorption/microbial anaerobic degradation risk management and control composite material and application thereof 浙江大学 2024-07-12 CN disclosed
CN-112209858-B Preparation method of 2- [ [ tri (hydroxymethyl) methyl ] amino ] ethanesulfonic acid 湖南韵邦生物医药有限公司 2022-11-01 CN disclosed
CN-114806914-A Yarrowia lipolytica for high yield of beta-carotene and application thereof 南京工业大学 2022-07-29 CN disclosed
CN-114634886-A Multifunctional microbial agent capable of degrading various halogenated organic pollutants simultaneously 河南科技大学 2022-06-17 CN disclosed
CN-114394680-A Application of microbial agent in degradation of various halogenated organic pollutants 河南科技大学 2022-04-26 CN disclosed
EP-2774630-B1 METHOD FOR PREPARING EDGE-RIGIDIZED ARTIFICIAL BIOLOGICAL VALVE SHANGHAI MICROPORT CARDIOFLOW MEDTECH CO LTD (CN) 2017-07-05 EP disclosed
EP-2774630-A1 METHOD FOR PREPARING EDGE-RIGIDIZED ARTIFICIAL BIOLOGICAL VALVE Shanghai MicroPort Medical (Group) Co., Ltd. (CN) 2014-09-10 EP disclosed
WO-2012103385-A2 BIOCATALYSTS SYNTHESIZING DEREGULATED CELLULASES QTEROS, INC. (US) 2012-08-02 WO disclosed
WO-2012068537-A2 NEW BIOCATALYSTS AND PRIMERS FOR PRODUCTION OF CHEMICALS QTEROS, INC. (US) 2012-05-24 WO disclosed
US-20120064592-A1 BIOCATALYSTS SYNTHESIZING DEREGULATED CELLULASES QTEROS, INC. (US) 2012-03-15 US disclosed
WO-2011072264-A2 METHODS AND COMPOSITIONS FOR BIOMASS TREATMENT QTEROS, INC. (US) 2011-06-16 WO disclosed