SCHEMBL4521923

SCHEMBL4521923

C[SiH](C)Oc1cc(C(C)(C)C)ccc1CCCBr

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTR1D P28221 4/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
HTR1A P08908 1/20 0.31
HTR1B P28222 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7586102 0.85 CYP2C19 (0.34) CYP1A2CYP2C19HTR1DCA1CA2
SCHEMBL8119764 0.84 CYP2C19 (0.38) CYP1A2CYP2C19HTR1DCA1CA2
SCHEMBL7592443 0.79 CA1 (0.40) CA1CA2CA9KDM4EATM
SCHEMBL8113705 0.78 KLF10 (0.39) CYP1A2CYP2C19HTR1DCA1CA2
SCHEMBL6760798 0.78 CYP2C19 (0.38) CYP1A2CYP2C19HTR1DCA1CA2
SCHEMBL4266306 0.77 NPSR1 (0.51) CYP2C19
SCHEMBL7999289 0.77 NPSR1 (0.40) CYP1A2CYP2C19HTR1DCA1CA2
SCHEMBL4261597 0.76 TP53 (0.41) CYP2C19HTR1DCA1CA2CA9
SCHEMBL7535667 0.75 NPSR1 (0.38) CYP2C19
SCHEMBL305273 0.73 CYP4F2 (0.44) CYP1A2CYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7498460-B2 Isophthalic acid derivatives BAYER HEALTHCARE AG (DE) 2009-03-03 US disclosed
EP-1572628-B1 ISOPHTALIC ACID DERIVATIVES BAYER HEALTHCARE AG (DE) 2007-07-25 EP disclosed
US-20060154912-A1 Isophtalic acid derivatives BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2006-07-13 US disclosed
EP-1572628-A1 ISOPHTALIC ACID DERIVATIVES Bayer HealthCare AG (DE) 2005-09-14 EP disclosed
WO-2004052839-A1 ISOPHTALIC ACID DERIVATIVES BAYER HEALTHCARE AG (DE) 2004-06-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060154912-A1 Isophtalic acid derivatives VHL, FABP3, CPT1A CYP1A2 96/4885CYP2C19 328/4885HTR1D 2426/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.