SCHEMBL4535758

SCHEMBL4535758

CCCN1CCN(C2(CNC(=O)c3cn(-c4ncccn4)c4nccc(Cl)c34)CCCCC2)CC1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCN4 Q9Y3Q4 7/20 0.50
HCN1 O60741 6/20 0.47
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
SLC6A9 P48067 9/20 0.45
OPRM1 P35372 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
TP53 P04637 1/20 0.43
P2RX7 Q99572 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4536437 0.94 HCN4 (0.54) HCN4HCN1ALDH1A1TSHRSLC6A9
SCHEMBL4350376 0.92 HCN4 (0.60) HCN4HCN1ALDH1A1TSHRSLC6A9
SCHEMBL13706858 0.92 HCN4 (0.60) HCN4HCN1ALDH1A1TSHRSLC6A9
SCHEMBL4537785 0.89 HCN4 (0.52) HCN4HCN1ALDH1A1TSHRSLC6A9
SCHEMBL13706860 0.88 HCN4 (0.55) HCN4HCN1ALDH1A1TSHRSLC6A9
SCHEMBL13706843 0.87 ALDH1A1 (0.56) HCN4ALDH1A1TSHRP2RX7
SCHEMBL13706906 0.87 HCN4 (0.51) HCN4HCN1ALDH1A1TSHRSLC6A9
SCHEMBL13706772 0.85 HCN4 (0.54) HCN4HCN1ALDH1A1TSHRSLC6A9
SCHEMBL13706774 0.84 HCN4 (0.55) HCN4HCN1ALDH1A1TSHRSLC6A9
SCHEMBL13706765 0.83 HCN4 (0.60) HCN4HCN1ALDH1A1TSHRSLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO claimed
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO disclosed