SCHEMBL4539019

SCHEMBL4539019

O=C(O)c1nccn1-c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.48
FDPS P14324 1/20 0.47
NR4A1 P22736 1/20 0.45
NR4A2 P43354 1/20 0.45
NOTUM Q6P988 1/20 0.44
ALDH1A1 P00352 5/20 0.43
CYP1A2 P05177 3/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2D6 P10635 3/20 0.43
CYP2C9 P11712 3/20 0.43
CYP2C19 P33261 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
POLB P06746 1/20 0.43
KDM4E B2RXH2 1/20 0.43
TSHR P16473 1/20 0.43
RAB9A P51151 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
NPC1 O15118 1/20 0.42
FGFR1 P11362 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27633478 0.89 ALDH1A1 (0.50) SMN1; SMN2FDPSNR4A1NR4A2NOTUM
SCHEMBL1345334 0.85 SMN1; SMN2 (0.46) SMN1; SMN2FDPSNR4A1NR4A2NOTUM
SCHEMBL7443999 0.85 SMN1; SMN2 (0.46) SMN1; SMN2FDPSNR4A1NR4A2NOTUM
SCHEMBL22290363 0.84 NR4A1 (0.49) SMN1; SMN2NR4A1NR4A2NOTUMALDH1A1
SCHEMBL23884809 0.81 ALDH1A1 (0.59) SMN1; SMN2NR4A1NR4A2ALDH1A1MEN1
SCHEMBL11177528 0.81 AKT1 (0.43) SMN1; SMN2FDPSNR4A1NR4A2NOTUM
SCHEMBL27807039 0.81 ALDH1A1 (0.48) SMN1; SMN2FDPSALDH1A1CYP1A2CYP3A4
SCHEMBL22290179 0.81 KMT2A (0.50) SMN1; SMN2FDPSNR4A2ALDH1A1CYP1A2
SCHEMBL25778550 0.80 KDM4E (0.66) SMN1; SMN2ALDH1A1CYP3A4CYP2C9POLB
SCHEMBL19651232 0.80 NR4A1 (0.42) NR4A1NR4A2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018064119-A1 CALPAIN MODULATORS AND THERAPEUTIC USES THEREOF BLADE THERAPEUTICS, INC. (US) 2018-04-05 WO disclosed
WO-2009117676-A2 NOVEL PIPERIDINE DERIVATIVES AS INHIBITORS OF STEAROYL-COA DESATURASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2009-09-24 WO disclosed
EP-0125783-B1 DOPAMINE-BETA-HYDROXYLASE INHIBITORS SMITHKLINE BECKMAN CORPORATION (US) 1989-01-04 EP disclosed