SCHEMBL4539673

SCHEMBL4539673

CCN1CC(=O)OC2(CCN(S(=O)(=O)c3ccc(-c4ccc5cc(F)cnc5c4)cc3)CC2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FASN P49327 4/20 0.44
ALDH1A1 P00352 3/20 0.36
CYP2D6 P10635 1/20 0.36
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
METAP2 P50579 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KDM2B Q8NHM5 1/20 0.34
LRRK2 Q5S007 2/20 0.34
SSTR5 P35346 1/20 0.33
KCNH2 Q12809 1/20 0.33
MTOR P42345 1/20 0.33
ADORA2A P29274 2/20 0.33
ADORA2B P29275 2/20 0.33
ADORA1 P30542 2/20 0.33
ADORA3 P0DMS8 1/20 0.33
PKM P14618 1/20 0.33
MEN1 O00255 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4540905 0.82 FASN (0.64) FASNALDH1A1METAP2SMN1; SMN2LRRK2
SCHEMBL4536294 0.77 FASN (0.56) FASNALDH1A1SMN1; SMN2LRRK2MTOR
SCHEMBL4540325 0.77 FASN (0.55) FASNALDH1A1KDM4EMETAP2SMN1; SMN2
SCHEMBL4541442 0.75 FASN (0.76) FASNALDH1A1SMN1; SMN2LRRK2MTOR
SCHEMBL4539655 0.70 FASN (0.62) FASNALDH1A1KDM4EMETAP2SMN1; SMN2
SCHEMBL4543103 0.68 FASN (0.73) FASNALDH1A1METAP2SMN1; SMN2PKM
SCHEMBL4539661 0.67 FASN (0.76) FASNALDH1A1CYP2D6SMN1; SMN2LRRK2
SCHEMBL4535806 0.66 FASN (0.51) FASNALDH1A1KDM4ESMN1; SMN2PKM
SCHEMBL4541212 0.66 FASN (0.55) FASNALDH1A1KDM4ESMN1; SMN2LRRK2
SCHEMBL4541537 0.66 FASN (0.54) FASNALDH1A1KDM4ESMN1; SMN2LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2637660-A1 FATTY ACID SYNTHASE INHIBITORS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2013-09-18 EP disclosed
WO-2012064642-A1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2012-05-18 WO disclosed