SCHEMBL4535806

SCHEMBL4535806

O=C1CN(C2CC2)CC2(CCN(S(=O)(=O)c3ccc(-c4ccc5ccccc5c4)cc3)CC2)O1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FASN P49327 4/20 0.51
ALDH1A1 P00352 6/20 0.45
KDM4E B2RXH2 4/20 0.45
PKM P14618 4/20 0.45
MCOLN3 Q8TDD5 3/20 0.42
LMNA P02545 3/20 0.42
TSHR P16473 3/20 0.40
MAPK1 P28482 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.39
USP2 O75604 2/20 0.39
HSD17B10 Q99714 2/20 0.39
HPGD P15428 1/20 0.39
HIF1A Q16665 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4561831 0.86 FASN (0.46) FASNALDH1A1KDM4EPKMMAPK1
SCHEMBL4538721 0.79 FASN (0.79) FASNALDH1A1KDM4EPKMMCOLN3
SCHEMBL4540739 0.78 CNR1 (0.38) FASNALDH1A1KDM4EPKML3MBTL1
SCHEMBL4538282 0.70 FASN (0.76) FASNALDH1A1PKMMAPK1MEN1
SCHEMBL22259570 0.70 FASN (0.58) FASNALDH1A1KDM4EPKMLMNA
SCHEMBL4540780 0.69 FASN (0.68) FASNALDH1A1KDM4EPKMMAPK1
SCHEMBL4540099 0.69 FASN (0.73) FASNALDH1A1KDM4EPKMLMNA
SCHEMBL4536291 0.68 MGLL (0.48) FASNALDH1A1KDM4EPKMMAPK1
SCHEMBL30754647 0.68 PKM (0.78) ALDH1A1PKMMCOLN3LMNATSHR
SCHEMBL4543035 0.68 FASN (1.00) FASNALDH1A1KDM4ELMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2637660-A1 FATTY ACID SYNTHASE INHIBITORS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2013-09-18 EP disclosed
WO-2012064642-A1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2012-05-18 WO disclosed